TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of steady-state expression of Raf-1 in MCF-7 breast cancer cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of steady-state expression of Raf-1 in MCF-7 breast cancer cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of steady-state expression of Raf-1 in MCF-7 breast cancer cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of DNA dependent protein kinase with hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.28E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.63E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.83E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.87E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.18E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.59E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.92E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department of Molecular Oncogenesis
Curated by ChEMBL
Department of Molecular Oncogenesis
Curated by ChEMBL
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 4.39E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 4.47E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 4.76E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.37E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.72E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.83E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 6.05E+4nMAssay Description:Inhibition of Hsp90 protein as degradation of HER2 kinase in SKBr3 cellsMore data for this Ligand-Target Pair