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Found 9 with Last Name = 'laplante' and Initial = 'p'
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220447(US10633379, Compound X | US9296741, 36)
Affinity DataIC50:  3nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataIC50:  5nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by chromatin/BRD4 displacement assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataIC50:  5nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataIC50:  5nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by chromatin/BRD4 displacement assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50:  30nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50510872(CHEMBL4303404)
Affinity DataIC50:  39nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50045000((NFLX)1-Ethyl-6-fluoro-4-oxo-7-piperazin-1-yl-1,4-...)
Affinity DataIC50:  980nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM76305(5-chloranylquinolin-8-ol | 5-chloro-8-quinolinol |...)
Affinity DataIC50:  6.47E+3nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  135nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair