TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 131nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 169nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 191nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 198nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 232nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 243nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 387nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 574nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of Tennessee
Curated by ChEMBL
University of Tennessee
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 655nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair