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Found 2294 with Last Name = 'ferguson' and Initial = 'r'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451823(CHEMBL2112840)
Affinity DataKi:  0.0600nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125686(2-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataKi:  0.170nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451820(CHEMBL3085267)
Affinity DataKi:  0.200nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451826(CHEMBL2112797)
Affinity DataKi:  0.210nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451822(CHEMBL2112839)
Affinity DataKi:  0.25nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451819(CHEMBL2079659)
Affinity DataKi:  0.280nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125687(2-[14-(6-carboxy-3,4,5-trihydroxytetrahydro-2H-2-p...)
Affinity DataKi:  0.600nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  0.780nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125689(6-[4-allyl-10-hydroxy-(5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  0.980nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451824(CHEMBL2092968)
Affinity DataKi:  1.20nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125680(3,4-dihydroxy-2-[10-hydroxy-4-methyl-(5R,13R,14S,1...)
Affinity DataKi:  1.40nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50370478(MORPHINE-6-GLUCURONIDE | Morphine 6-Glucuronide(Mi...)
Affinity DataKi:  1.5nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451825(CHEMBL2113393)
Affinity DataKi:  1.60nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451826(CHEMBL2112797)
Affinity DataKi:  2.5nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125688(3-hydroxy-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-...)
Affinity DataKi:  3.20nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451819(CHEMBL2079659)
Affinity DataKi:  3.20nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451823(CHEMBL2112840)
Affinity DataKi:  3.5nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451824(CHEMBL2092968)
Affinity DataKi:  4.80nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  4.80nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451822(CHEMBL2112839)
Affinity DataKi:  5.70nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125686(2-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataKi:  6.20nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451820(CHEMBL3085267)
Affinity DataKi:  10nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50370478(MORPHINE-6-GLUCURONIDE | Morphine 6-Glucuronide(Mi...)
Affinity DataKi:  26nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451821(CHEMBL3085275)
Affinity DataKi:  33nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125689(6-[4-allyl-10-hydroxy-(5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  37nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451825(CHEMBL2113393)
Affinity DataKi:  44nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125680(3,4-dihydroxy-2-[10-hydroxy-4-methyl-(5R,13R,14S,1...)
Affinity DataKi:  48nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125692(3,4,5-trihydroxy-6-[10-hydroxy-(5R,13R,14S,17R)-12...)
Affinity DataKi:  57nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125692(3,4,5-trihydroxy-6-[10-hydroxy-(5R,13R,14S,17R)-12...)
Affinity DataKi:  57nMAssay Description:mu-1 receptor binding affinity in rat brain by 3H [d-Ala2, d-Leu5] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125684(3,4,5-trihydroxy-6-[10-methoxy-4-methyl-(5R,13R,14...)
Affinity DataKi:  85nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125690(6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataKi:  168nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125690(6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataKi:  168nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125687(2-[14-(6-carboxy-3,4,5-trihydroxytetrahydro-2H-2-p...)
Affinity DataKi:  172nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125688(3-hydroxy-6-[10-hydroxy-4-methyl-(5R,13R,14S,17R)-...)
Affinity DataKi:  178nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50451821(CHEMBL3085275)
Affinity DataKi:  1.62E+3nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Ultrafine Ufc

Curated by ChEMBL
LigandPNGBDBM50125684(3,4,5-trihydroxy-6-[10-methoxy-4-methyl-(5R,13R,14...)
Affinity DataKi:  5.70E+3nMAssay Description:mu-2 receptor binding affinity in rat brain by 3H [d-Ala2, (N-Me)Phe4, Gly5-ol] enkephalin displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50437407(CHEMBL2408789 | US9023865, 6)
Affinity DataIC50:  0.152nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157165(US9023865, 11)
Affinity DataIC50:  0.152nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50437408(CHEMBL2408790 | US9023865, 2)
Affinity DataIC50:  0.152nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157642(US9023865, 483)
Affinity DataIC50:  0.152nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157225(US9023865, 71)
Affinity DataIC50:  0.159nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157778(US9023865, 619)
Affinity DataIC50:  0.159nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157343(US9023865, 184)
Affinity DataIC50:  0.171nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157706(US9023865, 547)
Affinity DataIC50:  0.184nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157739(US9023865, 580)
Affinity DataIC50:  0.193nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM272794(6-bromo-3-(2-methylpyridin-4-yl)-1,8-dihydro-7H-py...)
Affinity DataIC50:  0.200nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM272795(6-benzyl-3-(2-methylpyridin-4-yl)-1,8-dihydro-7H-p...)
Affinity DataIC50:  0.200nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM50437407(CHEMBL2408789 | US9023865, 6)
Affinity DataIC50:  0.204nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157164(US9023865, 10)
Affinity DataIC50:  0.215nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM157340(BDBM157741 | US9023865, 181)
Affinity DataIC50:  0.217nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
In DepthDetails US Patent
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