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TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221813(CHEMBL394602 | HO-LVA)
Affinity DataKi:  0.0320nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 384-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221813(CHEMBL394602 | HO-LVA)
Affinity DataKi:  0.0360nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 96-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075724(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-...)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075720((HO-LVA23)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-4-H...)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221815(4-({[(6-{N-[(1S)-5-amino-1-carbamoylpentyl]-1-[(3S...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.110nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.120nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.130nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.160nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075725(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(6C-...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075722(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50166224(CHEMBL410567 | Vasopressin Analogue)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against rat vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  0.180nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  0.190nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.200nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221813(CHEMBL394602 | HO-LVA)
Affinity DataKi:  0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221813(CHEMBL394602 | HO-LVA)
Affinity DataKi:  0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 384-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075728(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(6C-...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.240nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221813(CHEMBL394602 | HO-LVA)
Affinity DataKi:  0.280nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103475(Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe(I,N3)-NH2 | Pm...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  0.460nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.470nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 384-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103477(CHEMBL386180 | Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.650nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 96-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075721((LVA)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-phenylac...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50166219(CHEMBL264101 | Vasopressin Analogue)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  0.850nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50221815(4-({[(6-{N-[(1S)-5-amino-1-carbamoylpentyl]-1-[(3S...)
Affinity DataKi:  1.04nMAssay Description:Displacement of [3H]AVP from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50075721((LVA)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-phenylac...)
Affinity DataKi:  1.10nMAssay Description:The inhibition constant (Ki(nM)) of the compound was determined by displacement of [125I]- HO-LVA radiolabeled ligand using membranes of CHO cells of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50075724(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-...)
Affinity DataKi:  1.20nMAssay Description:The inhibition constant (Ki(nM)) of the compound was determined by displacement of [125I]- HO-LVA radiolabeled ligand using membranes of CHO cells of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075727(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Lys(5C-Rhm)-Pro...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  1.40nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  1.48nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 384-well plate membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50075722(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-...)
Affinity DataKi:  1.60nMAssay Description:The inhibition constant (Ki(nM)) of the compound was determined by displacement of [125I]- HO-LVA radiolabeled ligand using membranes of CHO cells of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50221816(5-({N-[(1S)-5-amino-1-carbamoylpentyl]-1-[(3S)-1-[...)
Affinity DataKi:  1.95nMAssay Description:Displacement of [3H]AVP from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50221816(5-({N-[(1S)-5-amino-1-carbamoylpentyl]-1-[(3S)-1-[...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103478(CHEMBL406670 | Pmp-Tyr(Me)-Ile-Thr-Asn-Cys-Pro-Orn...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50166225(CHEMBL410401 | Vasopressin Analogue)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50075720((HO-LVA23)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-4-H...)
Affinity DataKi:  2.70nMAssay Description:The inhibition constant (Ki(nM)) of the compound was determined by displacement of [125I]- HO-LVA radiolabeled ligand using membranes of CHO cells of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  3nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075729(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Lys(6C-Rhm)-Pro...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  4.80nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50075723(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Lys(5C-Flu)-Pro...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50075720((HO-LVA23)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-4-H...)
Affinity DataKi:  5.90nMAssay Description:Compound was tested for its ability to displace [125I]- HO-LVA ligand from human Vasopressin V1b receptor in the membranes of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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