TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Affinity of the Compound for Dopamine D1 receptor in rat striatal membrane was determined in vitro using Dopamine Antagonist [3H]SCH-23390 as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair