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Found 384 with Last Name = 'dunn' and Initial = 's'
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248829(CHEMBL4084229)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248829(CHEMBL4084229)
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM454169(BDBM50246180 | US10716791, Code KP-302)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246191(CHEMBL4089260)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246191(CHEMBL4089260)
Affinity DataKi:  7.10E+4nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM454162(BDBM50246174 | US10716791, Code KP-286)
Affinity DataKi:  8.80E+4nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50246191(CHEMBL4089260)
Affinity DataKi:  1.12E+5nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454169(BDBM50246180 | US10716791, Code KP-302)
Affinity DataKi:  1.55E+5nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM454169(BDBM50246180 | US10716791, Code KP-302)
Affinity DataKi:  1.80E+5nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.83E+5nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246193(CHEMBL4061099)
Affinity DataKi:  2.82E+5nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454164(BDBM50246192 | US10716791, Code KP-288)
Affinity DataKi:  3.53E+5nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50248829(CHEMBL4084229)
Affinity DataKi:  3.84E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  4.45E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM454165(BDBM50246195 | US10716791, Code KP-289)
Affinity DataKi:  4.88E+5nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM454162(BDBM50246174 | US10716791, Code KP-286)
Affinity DataKi:  5.54E+5nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM454164(BDBM50246192 | US10716791, Code KP-288)
Affinity DataKi:  5.91E+5nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50248824(CHEMBL4059499)
Affinity DataKi:  6.02E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248830(CHEMBL4089583)
Affinity DataKi:  6.32E+5nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248832(CHEMBL4084379)
Affinity DataKi:  7.14E+5nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454162(BDBM50246174 | US10716791, Code KP-286)
Affinity DataKi:  9.64E+5nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM454164(BDBM50246192 | US10716791, Code KP-288)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50246193(CHEMBL4061099)
Affinity DataKi:  1.09E+6nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248824(CHEMBL4059499)
Affinity DataKi:  1.43E+6nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM454165(BDBM50246195 | US10716791, Code KP-289)
Affinity DataKi:  1.84E+6nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50248814(CHEMBL4070114)
Affinity DataKi:  2.42E+6nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246193(CHEMBL4061099)
Affinity DataKi:  2.82E+6nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248830(CHEMBL4089583)
Affinity DataKi:  4.62E+6nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248831(CHEMBL4102346)
Affinity DataKi:  4.64E+6nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM454163(BDBM50246172 | US10716791, Code KP-287)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50246194(CHEMBL4062179 | US10716791, Example KP-316)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50246179(CHEMBL4081389)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246179(CHEMBL4081389)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246173(CHEMBL4082498)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246179(CHEMBL4081389)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50246173(CHEMBL4082498)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM454163(BDBM50246172 | US10716791, Code KP-287)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454163(BDBM50246172 | US10716791, Code KP-287)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))
Phoenix Molecular Designs

US Patent
LigandPNGBDBM286091((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...)
Affinity DataIC50:  0.300nMAssay Description:Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))
Phoenix Molecular Designs

US Patent
LigandPNGBDBM286091((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...)
Affinity DataIC50:  0.300nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Phoenix Molecular Design

US Patent
LigandPNGBDBM286091((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...)
Affinity DataIC50:  1.70nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Phoenix Molecular Design

US Patent
LigandPNGBDBM286091((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...)
Affinity DataIC50:  1.70nMAssay Description:Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Phoenix Molecular Design

US Patent
LigandPNGBDBM286091((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...)
Affinity DataIC50:  2nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Phoenix Molecular Design

US Patent
LigandPNGBDBM286091((R)¿N-(1-(4-aminobenzyl)-1H-pyrazol-4-yl)-9-methyl...)
Affinity DataIC50:  2nMAssay Description:Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50317833(3-methyl 5-(3-phenylbutyl)2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at rabbit Cav1.2 expressed in HEK293 cells assessed as inhibition of voltage pulse-induced calcium current by FLIPR calcium 4 ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Phoenix Molecular Design

US Patent
LigandPNGBDBM458758((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...)
Affinity DataIC50:  6nMAssay Description:Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Phoenix Molecular Design

US Patent
LigandPNGBDBM342166((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...)
Affinity DataIC50:  6nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50317821(3-(3,4-difluorobenzyl)5-methyl 2,6-dimethyl-4-(3-n...)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at rabbit Cav1.2 expressed in HEK293 cells assessed as inhibition of voltage pulse-induced calcium current by FLIPR calcium 4 ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))
Phoenix Molecular Designs

US Patent
LigandPNGBDBM342166((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...)
Affinity DataIC50:  8nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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