TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 637nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.25E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.54E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 5.21E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 2.85E+4nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: <0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: <0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: <0.200nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of HDAC2 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of HDAC1 (unknown origin) using compound purified by microgram-scale HPLC work-flowMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of HDAC3 (unknown origin) using compound purified by traditional preparative HPLC work-flowMore data for this Ligand-Target Pair