TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Competitive inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrateMore data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Inhibition of human RRM2 expressed in Escherichia coli BL21-codon plus(DE3) using [14C]-ADP as substrate after 3 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.72E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate by boronate affinity chromatographyMore data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 3.22E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 3.57E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 3.94E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 4.52E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 4.72E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 6.17E+4nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 7.01E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 8.68E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 9.41E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 9.52E+4nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of human RRM2 expressed in Escherichia coli BL21-codon plus(DE3) using [14C]-ADP as substrate after 3 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 1.31E+5nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 2.98E+5nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 6.87E+5nMAssay Description:Inhibition of human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL using [14C]-ADP as substrate after 3 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataIC50: 9.97E+5nMAssay Description:Inhibition of human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) using 14C-ADP as substrate by liquid scintillation c...More data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataKd: 1.08E+4nMAssay Description:Binding affinity to human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) by tryptophan fluorescence quenching assayMore data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataKd: 3.56E+4nMAssay Description:Binding affinity to human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) by tryptophan fluorescence quenching assayMore data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataKd: 3.70E+4nMAssay Description:Binding affinity to human RRM1 expressed in Escherichia coli BL21-codon plus(DE3)-RIL by fluorescence spectrophotometric methodMore data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataKd: 9.68E+3nMAssay Description:Binding affinity to human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) by tryptophan fluorescence quenching assayMore data for this Ligand-Target Pair
TargetRibonucleoside-diphosphate reductase large subunit(Homo sapiens (Human))
Case Western Reserve University
Curated by ChEMBL
Case Western Reserve University
Curated by ChEMBL
Affinity DataKd: 5.53E+4nMAssay Description:Binding affinity to human ribonucleotide reductase M1 subunit expressed in Escherichia coli BL21 (DE3) by tryptophan fluorescence quenching assayMore data for this Ligand-Target Pair