Affinity DataKi: 0.300nMAssay Description:Competitive inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Competitive inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.15E+3nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.30E+3nMAssay Description:In vitro binding affinity towards melanocortin 4 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL