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Found 168 with Last Name = 'tsujino' and Initial = 't'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296870((1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296879((4,4-diphenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-m...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296884((1-((1R,4R)-2,2-dimethyl-4-((R)-1-p-tolylethylamin...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296885(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296873(1'-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296881((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296877(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296883((1-((1R,4R)-4-((R)-1-(4-chlorophenyl)ethylamino)-2...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296878(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296876((4-(6-chloropyridin-3-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296872(3-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296880((1-((1R,4R)-2,2-dimethyl-4-((S)-2,2,2-trifluoro-1-...)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296882((1-((1R,4R)-4-((R)-1-(4-fluorophenyl)ethylamino)-2...)
Affinity DataKi:  44nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296871(1-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296875(CHEMBL556915 | N-(4-((1R,4R)-4-((R)-1-(4-methoxyph...)
Affinity DataKi:  48nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296874(CHEMBL561193 | N-(4-((1R,4R)-4-((R)-1-(4-methoxyph...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296894(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296891((1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296888((1-((1R,4R)-2,2-dimethyl-4-((R)-1-phenylethylamino...)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296886((1-((1R,4R)-4-((R)-1-(3-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296893(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  330nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296889((1-((1R,4R)-4-(4-methoxybenzylamino)-2,2-dimethylc...)
Affinity DataKi:  470nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296887((1-((1R,4R)-4-((R)-1-(2-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  790nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296895((4-(1,3,4-oxadiazol-2-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataKi:  890nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296890((1-((1R,4R)-4-((S)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296892(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296002(CHEMBL564536 | isopropyl 3-chloro-5-(1-(6-(2-(5-et...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]PYY from human recombinant NPY Y1 receptor expressed in CHO cells assessed as inhibition of [35S]GTPgammaS binding by scinitill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297965((R)-3-(1-(2-chloro-4-(hydroxymethyl)phenyl)ethoxy)...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297962((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(imidazo[1,2-a]...)
Affinity DataIC50:  7nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297966((R)-3-(1-(2-chlorophenyl)ethoxy)-5-(6-(hydroxymeth...)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296876((4-(6-chloropyridin-3-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297985((R)-3-(1-(4-((tert-butylamino)methyl)-2-(difluorom...)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296873(1'-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297971((R)-3-(1-(2-chloro-4-((cyclopropylamino)methyl)phe...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297981((R)-3-(1-(2-chloro-4-((3-oxopiperazin-1-yl)methyl)...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297977((R)-3-(1-(2-chloro-4-((4-fluoropiperidin-1-yl)meth...)
Affinity DataIC50:  13nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296877(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296874(CHEMBL561193 | N-(4-((1R,4R)-4-((R)-1-(4-methoxyph...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296879((4,4-diphenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-m...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297982(3-{(R)-1-[2-Chloro-4-(1,1-dioxo-1lambda*6*-thiomor...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297967((R)-3-(1-(2-chloro-4-((methylamino)methyl)phenyl)e...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296870((1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296878(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296872(3-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297978((R)-3-(1-(2-chloro-4-((4-methylpiperazin-1-yl)meth...)
Affinity DataIC50:  17nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297975((R)-3-(1-(2-chloro-4-((3-hydroxypropylamino)methyl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297980(3-((1R)-1-(2-chloro-4-((3-hydroxypyrrolidin-1-yl)m...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297984((R)-3-(1-(4-((tert-butylamino)methyl)-2-(difluorom...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297973((R)-3-(1-(4-((tert-butylamino)methyl)-2-chlorophen...)
Affinity DataIC50:  21nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297969((R)-3-(1-(2-chloro-4-((ethylamino)methyl)phenyl)et...)
Affinity DataIC50:  21nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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