Affinity DataKi: 0.400nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.01nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 1.61nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 2.96nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 4.77nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights
Curated by ChEMBL
University Heights
Curated by ChEMBL
Affinity DataKi: 9.32nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair