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Found 54 with Last Name = 'gioannini' and Initial = 'tl'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataIC50:  1.5nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  2nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  2nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225681(CHEMBL611395)
Affinity DataIC50:  2.30nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021257(2-[11,15-dimethoxy-3-methyl-(14R)-13-oxa-3-azahexa...)
Affinity DataIC50:  2.5nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225681(CHEMBL611395)
Affinity DataIC50:  3.5nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  4nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  4nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225690(CHEMBL610808)
Affinity DataIC50:  6nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225684(CHEMBL610611)
Affinity DataIC50:  6nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021255(2-[11,15-dimethoxy-3-methyl-(1R,14R,15R)-13-oxa-3-...)
Affinity DataIC50:  6.40nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225683(CHEMBL610807)
Affinity DataIC50:  7nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225685(CHEMBL175344)
Affinity DataIC50:  8nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225690(CHEMBL610808)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225692(CHEMBL610612)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021258(4-(4-allyloxyphenyl)-2-(11,15-dimethoxy-3-methyl-1...)
Affinity DataIC50:  10nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225692(CHEMBL610612)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225683(CHEMBL610807)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  12.5nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  12.5nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  13nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  13nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225682(CHEMBL174530)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225693(CHEMBL369657)
Affinity DataIC50:  30nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  35nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  35nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021257(2-[11,15-dimethoxy-3-methyl-(14R)-13-oxa-3-azahexa...)
Affinity DataIC50:  38nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225688(CHEMBL611391)
Affinity DataIC50:  40nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021255(2-[11,15-dimethoxy-3-methyl-(1R,14R,15R)-13-oxa-3-...)
Affinity DataIC50:  50nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225689(CHEMBL611392)
Affinity DataIC50:  50nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225685(CHEMBL175344)
Affinity DataIC50:  60nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225686(CHEMBL367540)
Affinity DataIC50:  70nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225688(CHEMBL611391)
Affinity DataIC50:  70nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021258(4-(4-allyloxyphenyl)-2-(11,15-dimethoxy-3-methyl-1...)
Affinity DataIC50:  84nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021253(7alpha-[(1R)-1-Hydroxy1-methyl-3-[4-[3-(bromomercu...)
Affinity DataIC50:  95nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225689(CHEMBL611392)
Affinity DataIC50:  100nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021254(7alpha-[(1R)-1-Hydroxy1-methyl-3-[4-[3-(bromomercu...)
Affinity DataIC50:  100nMAssay Description:Evaluated for the inhibition of [3H]naltrexone binding to Opioid receptor mu 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021254(7alpha-[(1R)-1-Hydroxy1-methyl-3-[4-[3-(bromomercu...)
Affinity DataIC50:  100nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  115nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  115nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225682(CHEMBL174530)
Affinity DataIC50:  200nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225691(CHEMBL174268)
Affinity DataIC50:  200nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  250nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50021253(7alpha-[(1R)-1-Hydroxy1-methyl-3-[4-[3-(bromomercu...)
Affinity DataIC50:  250nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  250nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225693(CHEMBL369657)
Affinity DataIC50:  500nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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