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Found 644 with Last Name = 'burkholder' and Initial = 'tp'
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063687(CHEMBL3397339)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063689(CHEMBL3397337)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063755(CHEMBL3397341)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063688(CHEMBL3397338)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063686(CHEMBL3397340)
Affinity DataKi:  0.180nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063690(CHEMBL3397336)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063754(CHEMBL3397342)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063689(CHEMBL3397337)
Affinity DataKi:  0.350nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063691(CHEMBL3397335)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063687(CHEMBL3397339)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063755(CHEMBL3397341)
Affinity DataKi:  0.510nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063752(CHEMBL3397343)
Affinity DataKi:  0.540nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063751(CHEMBL3397344)
Affinity DataKi:  0.640nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Bos taurus)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Bos taurus)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  0.960nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063693(CHEMBL3397333)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  1.02nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063692(CHEMBL3397334)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063690(CHEMBL3397336)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063750(CHEMBL3397345)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50030178((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataKi:  1.49nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(HAMSTER)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063688(CHEMBL3397338)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  2.12nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063686(CHEMBL3397340)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  2.99nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063695(CHEMBL3397346)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  3.11nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50030178((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataKi:  3.13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81944(CAS_86933-75-7 | NKB | NSC_5311312 | neuromedin K)
Affinity DataKi:  3.54nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  3.69nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50290297(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  5.88nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(HAMSTER)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  6.98nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50290297(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  7.07nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(HAMSTER)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  7.32nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063691(CHEMBL3397335)
Affinity DataKi:  7.70nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  7.93nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063694(CHEMBL3397347)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRbeta expressed in human Hela cell lysate measured after overnight incubation by competi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50029885((3aR,7aR)-2-[1-Imino-2-(2-methoxy-phenyl)-ethyl]-7...)
Affinity DataKi:  8.29nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Bos taurus)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  8.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  8.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Bos taurus)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  8.49nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063754(CHEMBL3397342)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50279944((R)-2-(2-Carboxymethyl-3-oxo-2,3,4,5-tetrahydro-1H...)
Affinity DataKi:  10nMAssay Description:Inhibitory constant of the compound was tested angiotensin converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50063693(CHEMBL3397333)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-L-3,5,3'-triiodothyronine from human TRalpha expressed in human Hela cell lysate measured after overnight incubation by compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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