Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of adenosine deaminase assessed as conversion of adenosine to inosineMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.05E+4nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 5.05E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.67E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: 5.95E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 5.95E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.21E+4nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 8.09E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: 8.16E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 8.29E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 9.90E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences
Curated by ChEMBL
Swedish University Agricultural Sciences
Curated by ChEMBL
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair