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Found 57 with Last Name = 'mcbrayer' and Initial = 'tr'
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432235(CHEMBL2347323)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387086(CHEMBL2047191)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50356463(CHEMBL1911841)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of adenosine deaminase assessed as conversion of adenosine to inosineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432236(CHEMBL2347159)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Rfs Pharma

Curated by ChEMBL
LigandPNGBDBM50484706(CHEMBL1950241)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Rfs Pharma

Curated by ChEMBL
LigandPNGBDBM50484704(CHEMBL1950242)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432234(CHEMBL2347328)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432233(CHEMBL2347337)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432234(CHEMBL2347328)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Ureaplasma parvum)
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387085(CHEMBL2047188)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Rfs Pharma

Curated by ChEMBL
LigandPNGBDBM50484705(CHEMBL1950240)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432233(CHEMBL2347337)
Affinity DataIC50:  3.12E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317617(3'-(4-(4-Fluorophenyl)-1,2,3-triazole-1-yl)-2'-deo...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432235(CHEMBL2347323)
Affinity DataIC50:  5.05E+4nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432235(CHEMBL2347323)
Affinity DataIC50:  5.05E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Rfs Pharma

Curated by ChEMBL
LigandPNGBDBM50478972(2''C-Me-CTP | CHEMBL223585)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of Hepatitis C virus NS5B Cdelta 21 RNA dependent RNA polymerase S282T mutant expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50314841(3'-(4-(2-Pyridine)-1,2,3-triazole-1-yl)-2'-deoxyth...)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432233(CHEMBL2347337)
Affinity DataIC50:  5.67E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50:  5.95E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50:  5.95E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317618(3'-(4-(2-Phenyl-ethyl)-1,2,3-triazole-1-yl)-2'-deo...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432234(CHEMBL2347328)
Affinity DataIC50:  6.21E+4nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Ureaplasma parvum)
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317617(3'-(4-(4-Fluorophenyl)-1,2,3-triazole-1-yl)-2'-deo...)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Ureaplasma parvum)
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50314837(3'-(4-Benzyl-1,2,3-triazol-1-yl)-3'-deoxy-beta-D-t...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50314837(3'-(4-Benzyl-1,2,3-triazol-1-yl)-3'-deoxy-beta-D-t...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432235(CHEMBL2347323)
Affinity DataIC50:  8.09E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387085(CHEMBL2047188)
Affinity DataIC50:  8.16E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432234(CHEMBL2347328)
Affinity DataIC50:  8.29E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317619(3'-(4-Pentyl-1,2,3-triazol-1-yl)-3'-deoxythymidine...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50314836(3'-(4-Phenyl-1,2,3-triazol-1-yl)-3'-deoxythymidine...)
Affinity DataIC50:  9.90E+4nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432236(CHEMBL2347159)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432233(CHEMBL2347337)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432236(CHEMBL2347159)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387086(CHEMBL2047191)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387086(CHEMBL2047191)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387085(CHEMBL2047188)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387086(CHEMBL2047191)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387085(CHEMBL2047188)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50432236(CHEMBL2347159)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317622(3'-(4-(3-Chloro-propyl)-1,2,3-triazol-1-yl)-3'-deo...)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317620(3'-(4-tert-Butyl-1,2,3-triazol-1-yl)-3'-deoxythymi...)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Ureaplasma parvum)
Swedish University Agricultural Sciences

Curated by ChEMBL
LigandPNGBDBM50317618(3'-(4-(2-Phenyl-ethyl)-1,2,3-triazole-1-yl)-2'-deo...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of Ureaplasma parvum thymidine kinase by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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