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Found 99 with Last Name = 'gräfe' and Initial = 'u'
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216095(5-(4-cyclohexylthiosemicarbazono)methyl-2-hydroxy-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50359629(TROLOX)
Affinity DataIC50:  130nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50359629(TROLOX)
Affinity DataIC50:  150nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216114(3-(4-cyclohexylthiosemicarbazono)methyl-2-hydroxy-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216102(3-(4-cyclohexylthiosemicarbazono)methyl-4-hydroxy-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216115(3-((cyclohexylaminocarbonothioyl)hydrazono]methyl)...)
Affinity DataIC50:  460nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216115(3-((cyclohexylaminocarbonothioyl)hydrazono]methyl)...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50371115(CHEMBL232615)
Affinity DataIC50:  630nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216125(6-(4-cyclohexylthiosemicarbazono)methyl-2-hydroxy-...)
Affinity DataIC50:  730nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216126(3-(1H-tetrazol-5-yl)-benzaldehyde cyclohexylthiose...)
Affinity DataIC50:  810nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216119(3-(4-cyclohexylthiosemicarbazono)methylbenzoic aci...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112868(3-((N-cyclohexyl-N-methylaminocarbonothioyl)hydraz...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112848(3-((cycloheptylaminocarbonothioyl)hydrazono]methyl...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM35440(ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of Xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216127(4-(4-cyclohexylthiosemicarbazono)methyl-phenol | C...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216094((E,Z)-2-(4-cyclohexylthiosemicarbazono)methyl-6-hy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50051829(4-methyl-2-oxo-2H-chromen-7-yl sulfamate | CHEMBL1...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM13058(6-oxo-6,7,8,9,10,11-hexahydrocyclohepta[c]chromen-...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112851(3-((cyclopentylaminocarbonothioyl)hydrazono]methyl...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216099(CHEMBL389867 | sodium 2-(4-cyclohexylthiosemicarba...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216129(3-(4-cycloheptylthiosemicarbazono)methyl-benzoic a...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216118(3-(4-cyclohexylthiosemicarbazono)methyl-phenol | C...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216100(2-(4-cyclohexylthiosemicarbazono)methylbenzoic aci...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112862(3-(((4-methyl-cyclohexyl)aminocarbonothioyl)hydraz...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216109(2-(4-cyclohexylthiosemicarbazono)methyl-6-hydroxy-...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216116(6-(4-cyclohexylthiosemicarbazono)methyl-2,3-dihydr...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216121(CHEMBL389890 | sodium 3-(4-cyclohexylthiosemicarba...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50371115(CHEMBL232615)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112849(3-((phenylaminocarbonothioyl)hydrazono]methyl)-1,9...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216123(3-(4-cyclohexylthiosemicarbazono)methyl-4-hydroxy-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112853(3-((Butylaminocarbonothioyl)hydrazono]methyl)-1,9,...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112865(3-((N-piperidinyl-aminocarbonothioyl)hydrazono]met...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112876(3-((N-cyclohexyl-aminocarbonoyl)hydrazono]methyl)-...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112873(1,9,11,14-Tetrahydroxy-7-methoxy-10-methyl-8,13-di...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112875(3-((Hexylaminocarbonothioyl)hydrazono]methyl)-1,9,...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216096(2-(4-cyclohexylthiosemicarbazono)methyl-phenol | C...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112852(3-((Heptylaminocarbonothioyl)hydrazono]methyl)-1,9...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50269144(10-hydroxy-18-methoxybetaenone | CHEMBL498247)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112855(3-((Isobutylaminocarbonothioyl)hydrazono]methyl)-1...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Heinrich-Heine-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50269144(10-hydroxy-18-methoxybetaenone | CHEMBL498247)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112856(3-(((4-methyl-phenyl)aminocarbonothioyl)hydrazono]...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216113(3-(4-hexylthiosemicarbazono)methyl-benzoic acid | ...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112863(3-((Pentylaminocarbonothioyl)hydrazono]methyl)-1,9...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216110(2-(4-cyclohexylthiosemicarbazono)methyl-benzoic ac...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50216108(2-(4-cycloheptylthiosemicarbazono)methyl-benzoic a...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Estrone sulfatase in human placental microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDehydrogenase/reductase SDR family member 9(Homo sapiens (Human))
Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of 3alphaHSDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Institute For Natural Products Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM50112850(3-((cyclooctylaminocarbonothioyl)hydrazono]methyl)...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory activity againist Estrone sulfatase from MCF-7 cells (placental microsomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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