Compile Data Set for Download or QSAR
maximum 50k data
Found 138 with Last Name = 'guerrant' and Initial = 'w'
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478829(6-(6-Methoxynaphthalyl)Triazolylhexahydroxamic Aci...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478811(6-(3-Biphenyl)Triazolylhexahydroxamic Acid | CHEMB...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27188(triazole-linked clarithromycin-based compound, 24d)
Affinity DataIC50:  1.90nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478823(6-(2-Quinolyl)Triazolylhexahydroxamic Acid | CHEMB...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478814(6-(4-Anisolyl)Triazolylhexahydroxamic Acid | CHEMB...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478832(6-(4-Pyridylphenyl)Triazolylhexahydroxamic Acid | ...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50481553(7-(2-Tolyl)Triazolylheptahydroxamamic Acid | CHEMB...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27187(triazole-linked clarithromycin-based compound, 24c)
Affinity DataIC50:  4.10nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478819(6-(4-Anilyl)Triazolylhexahydroxamic Acid | CHEMBL4...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  5nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478810(7-(3-Biphenyl)Triazolylheptahydroxamic Acid | CHEM...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM50382632(CHEMBL2023529)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC1 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478820(7-(Phenyl)Triazolylheptahydroxamic Acid | CHEMBL47...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Plasmodium falciparum (isolate 3D7))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50324111(CHEMBL1214760)
Affinity DataIC50:  10nMAssay Description:Inhibition of Plasmodium falciparum HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27180(7-{4-[4-({[(2S,3R,4S,6R)-2-{[(2R,3S,4R,5R,8R,10R,1...)
Affinity DataIC50:  10.6nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM50382631(CHEMBL2023530)
Affinity DataIC50:  11nMAssay Description:Inhibition of HDAC1 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27179(triazole-linked azithromycin-based compound, 16c)
Affinity DataIC50:  13.9nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478825(6-(3-Anisolyl)Triazolylhexahydroxamic Acid | CHEMB...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478828(6-(Phenyl)Triazolylhexahydroxamic Acid | CHEMBL478...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478808(7-(6-Methoxynaphthalyl)Triazolylheptahydroxamic Ac...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50481551(CHEMBL590567)
Affinity DataIC50:  16nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478830(7-(4-Pyridylphenyl)Triazolylheptahydroxamic Acid |...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478815(CHEMBL478310)
Affinity DataIC50:  17nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50382631(CHEMBL2023530)
Affinity DataIC50:  19nMAssay Description:Inhibition of HDAC6 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50382632(CHEMBL2023529)
Affinity DataIC50:  20nMAssay Description:Inhibition of HDAC6 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50382634(CHEMBL2023526)
Affinity DataIC50:  20nMAssay Description:Inhibition of HDAC6 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478831(7-(2-Pyridyl)Triazolylheptahydroxamic Acid | CHEMB...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  27nMAssay Description:Inhibition of HDAC6 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  27nMAssay Description:Inhibition of HDAC6 in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50382633(CHEMBL2023528)
Affinity DataIC50:  30nMAssay Description:Inhibition of HDAC6 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478816(6-(3-Tolyl)Triazolylhexahydroxamic Acid | CHEMBL51...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478812(6-(2-Thiopyl)Triazolylhexahydroxamic Acid | CHEMBL...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50491819(CHEMBL2386908)
Affinity DataIC50:  36nMAssay Description:Inhibition of HDAC6 in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Plasmodium falciparum (isolate 3D7))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50324110(CHEMBL1214759)
Affinity DataIC50:  36nMAssay Description:Inhibition of Plasmodium falciparum HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27185(triazole-linked clarithromycin-based compound, 24a)
Affinity DataIC50:  37nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM50491817(CHEMBL2386912)
Affinity DataIC50:  37nMAssay Description:Inhibition of HDAC1 in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HDAC1 in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HDAC1 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase(Plasmodium falciparum (isolate 3D7))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50324114(CHEMBL1214761)
Affinity DataIC50:  40nMAssay Description:Inhibition of Plasmodium falciparum HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50491820(CHEMBL2386907)
Affinity DataIC50:  42nMAssay Description:Inhibition of HDAC6 in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478826(6-(4-Tolyl)Triazolylhexahydroxamic Acid | CHEMBL50...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27186(triazole-linked clarithromycin-based compound, 24b)
Affinity DataIC50:  44.3nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM50382634(CHEMBL2023526)
Affinity DataIC50:  47nMAssay Description:Inhibition of HDAC1 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM50491819(CHEMBL2386908)
Affinity DataIC50:  50nMAssay Description:Inhibition of HDAC1 in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50478824(6-(4-Biphenyl)Triazolylhexahydroxamic Acid | CHEMB...)
Affinity DataIC50:  52nMAssay Description:Inhibition of human HDAC in HeLa cells by flour de lys assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM50382633(CHEMBL2023528)
Affinity DataIC50:  54nMAssay Description:Inhibition of HDAC1 in human HeLa cell nuclear extract using Fluor de Lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50481556(9-(Phenyl)Triazolylnonahydroxamic Acid | CHEMBL591...)
Affinity DataIC50:  55nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extracts after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Georgia Institute of Technology

LigandPNGBDBM27189(triazole-linked clarithromycin-based compound, 24e)
Affinity DataIC50:  55.6nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Georgia Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50491817(CHEMBL2386912)
Affinity DataIC50:  56nMAssay Description:Inhibition of HDAC in human HeLa cells using Fluor-de-Lys as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 138 total ) | Next | Last >>
Jump to: