Affinity DataKi: 0.0280nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nM ΔG°: -54.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nM ΔG°: -51.9kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nM ΔG°: -49.7kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair