Affinity DataKi: 0.00500nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2.89nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 5.85nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 9.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition against Opioid receptor delta 1 using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [125I]IMPY from human beta amyloid plaque in brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 1.18E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 3.92E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences and Peking Union Medical College
Curated by ChEMBL
Affinity DataKi: 8.87E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
The Hong Kong Polytechnic University
Curated by ChEMBL
The Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Inhibition of wild type N-terminal His6-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21 assessed as inhibition constant using n...More data for this Ligand-Target Pair