Affinity DataKi: 1nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity for Bradykinin receptor B2 expressed in COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of aurora-A (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T
Curated by ChEMBL
Heinrich Heine Universit£T
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of aurora-B (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of SAK (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of aurora-A (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of COT (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CDK4/cyclin-D1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of INSR (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CDK4/cyclin-D1 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of COT (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of VEGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CDK2/cyclin-A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of aurora-B (unknown origin)More data for this Ligand-Target Pair
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of ARK5 (unknown origin)More data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of aurora-A (unknown origin)More data for this Ligand-Target Pair
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ARK5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of SAK (unknown origin)More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Heinrich-Heine University
Curated by ChEMBL
Heinrich-Heine University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of AKT1 (unknown origin)More data for this Ligand-Target Pair