Affinity DataIC50: 56nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 154nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 159nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 192nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 203nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 305nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 325nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 337nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 594nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 663nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 909nMAssay Description:Inhibitory concentration against serine protease chymase was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.96E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.44E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.57E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.59E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.21E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.28E+3nMAssay Description:Antagonist activity against human S1P1 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.18E+3nMAssay Description:Antagonist activity against human S1P1 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.64E+3nMAssay Description:Antagonist activity against human S1P1 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.75E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.74E+3nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+4nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.16E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Antagonist activity against human S1P3 receptor assessed as inhibition of S1P-induced intracellular calcium mobilization in CHO-K1 cellsMore data for this Ligand-Target Pair