Affinity DataKi: 0.330nM ΔG°: -54.1kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.470nM ΔG°: -53.2kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.560nM ΔG°: -52.8kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nM ΔG°: -51.8kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.910nM ΔG°: -51.6kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.01nMAssay Description:compound was tested in vitro for inhibition of serine protease thrombin(FIIa).More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.13nM ΔG°: -51.1kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nM ΔG°: -50.7kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nM ΔG°: -50.2kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.68nM ΔG°: -50.1kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 2nM ΔG°: -50.5kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.29nM ΔG°: -49.3kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.46nM ΔG°: -49.1kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nM ΔG°: -48.9kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.01nM ΔG°: -48.6kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cerebral membrane after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.73nM ΔG°: -48.1kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 3.80nM ΔG°: -48.9kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nM ΔG°: -48.0kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.99nM ΔG°: -47.9kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.05nM ΔG°: -47.9kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 4.99nM ΔG°: -47.4kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.02nM ΔG°: -47.4kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.18nM ΔG°: -47.3kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.20nM ΔG°: -47.3kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.23nM ΔG°: -47.3kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.28nM ΔG°: -47.2kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.34nM ΔG°: -47.2kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.36nM ΔG°: -47.2kJ/moleT: 2°CAssay Description:Binding assay of opioid receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
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