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Found 49 with Last Name = 'chang' and Initial = 'yj'
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321752(5-Chloro-2-(2-methoxyphenyl)-4H-benzo[d][1,3]oxazi...)
Affinity DataIC50:  15.4nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321750(5-Chloro-2-(2-bromophenyl)-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50:  24.8nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321749(5-Chloro-2-(2-chlorophenyl)-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50:  28.7nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321750(5-Chloro-2-(2-bromophenyl)-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50:  29.5nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321749(5-Chloro-2-(2-chlorophenyl)-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50:  30.7nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321748(5-Chloro-2-(2-fluorophenyl)-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50:  30.8nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321752(5-Chloro-2-(2-methoxyphenyl)-4H-benzo[d][1,3]oxazi...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321751(5-Chloro-2-(2-methylphenyl)-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50:  48.8nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321748(5-Chloro-2-(2-fluorophenyl)-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50:  52.7nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321751(5-Chloro-2-(2-methylphenyl)-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50:  57.1nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435554(CHEMBL2392817)
Affinity DataIC50:  58nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50299853(1-(3,4-Dimethoxyphenyl)-3-(3-(5-methyl-1H-imidazol...)
Affinity DataIC50:  119nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435549(CHEMBL2392800)
Affinity DataIC50:  123nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435533(CHEMBL2392794)
Affinity DataIC50:  158nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435561(CHEMBL2392810)
Affinity DataIC50:  185nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435558(CHEMBL2392814)
Affinity DataIC50:  208nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321747(7-Chloro-2-(2-methoxyphenyl)-4H-benzo[d][1,3]oxazi...)
Affinity DataIC50:  222nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435547(CHEMBL2392803)
Affinity DataIC50:  239nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435532(CHEMBL2392778)
Affinity DataIC50:  293nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435539(CHEMBL2392786)
Affinity DataIC50:  329nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435534(CHEMBL2392793)
Affinity DataIC50:  337nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435529(CHEMBL2392783)
Affinity DataIC50:  375nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435546(CHEMBL2392804)
Affinity DataIC50:  381nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435559(CHEMBL2392813)
Affinity DataIC50:  405nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435560(CHEMBL2392812)
Affinity DataIC50:  437nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435536(CHEMBL2392789)
Affinity DataIC50:  453nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435543(CHEMBL2392807)
Affinity DataIC50:  461nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435545(CHEMBL2392805)
Affinity DataIC50:  463nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435542(CHEMBL2392808)
Affinity DataIC50:  475nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435557(CHEMBL2390975)
Affinity DataIC50:  479nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435553(CHEMBL2392796)
Affinity DataIC50:  482nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435537(CHEMBL2392788)
Affinity DataIC50:  488nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435556(CHEMBL2392815)
Affinity DataIC50:  492nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435535(CHEMBL2392791)
Affinity DataIC50:  518nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435551(CHEMBL2392798)
Affinity DataIC50:  519nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435541(CHEMBL2392809)
Affinity DataIC50:  524nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435530(CHEMBL2392782)
Affinity DataIC50:  546nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50321747(7-Chloro-2-(2-methoxyphenyl)-4H-benzo[d][1,3]oxazi...)
Affinity DataIC50:  612nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435544(CHEMBL2392806)
Affinity DataIC50:  711nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435531(CHEMBL2392779)
Affinity DataIC50:  768nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435552(CHEMBL2392797)
Affinity DataIC50:  788nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435550(CHEMBL2392799)
Affinity DataIC50:  812nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435555(CHEMBL2392816)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435540(CHEMBL2392785)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435538(CHEMBL2392787)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435548(CHEMBL2392802)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435528(CHEMBL2392784)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50171289(Benzenemethanesulfonyl fluoride | CHEMBL190503 | P...)
Affinity DataIC50:  5.22E+4nMAssay Description:Inhibition of human leukocyte elastase after 2 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50171289(Benzenemethanesulfonyl fluoride | CHEMBL190503 | P...)
Affinity DataIC50:  9.52E+4nMAssay Description:Inhibition of human neutrophil elastase after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed