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Found 39 with Last Name = 'ashendel' and Initial = 'cl'
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217039(CHEMBL420938)
Affinity DataIC50:  300nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217036(CHEMBL74983)
Affinity DataIC50:  700nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217032(CHEMBL76100)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230709(CHEMBL295954)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217040(CHEMBL73495)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230703(CHEMBL296591)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230702(CHEMBL48695)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230712(CHEMBL52232)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230714(CHEMBL48551)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230705(CHEMBL49951)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230711(CHEMBL441041)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50478491(GOB C)
Affinity DataIC50:  7.68E+3nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230704(CHEMBL416830)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230713(CHEMBL301124)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50478490(CHEMBL476674)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230701(CHEBI:73067 | Palmitoyl-carnitine)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217033(CHEMBL308288)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataIC50:  4.96E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM79181(10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoro...)
Affinity DataIC50:  7.36E+4nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50131698((Z)-resveratrol | 5-[(1Z)-2-(4-hydroxyphenyl)ethen...)
Affinity DataIC50:  1.31E+5nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50230710(CHEMBL49275)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataIC50:  1.75E+5nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284164((S)-2-Hexadecyl-2-hydroxy-4,4-dimethyl-morpholin-4...)
Affinity DataIC50:  2.35E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II); Range = 32-235 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217037(CHEMBL72370)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  3.05E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal carnitine O-octanoyltransferase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  4.75E+5nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217024(CHEMBL309186)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM79181(10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoro...)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM60919((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[3-[(E)-2-(4-...)
Affinity DataIC50:  5.12E+5nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50478492(CHEBI:76155 | Z-PICEID)
Affinity DataIC50:  5.12E+5nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal carnitine O-octanoyltransferase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  9.12E+5nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217041(CHEMBL73197)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217034(CHEMBL310913)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217042(CHEMBL75706)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217038(CHEMBL76469)
Affinity DataIC50: >4.00E+6nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50217035(CHEBI:87611 | CHEMBL72211 | Thiophene-3-Carbaldehy...)
Affinity DataIC50: >4.00E+6nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal carnitine O-octanoyltransferase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284164((S)-2-Hexadecyl-2-hydroxy-4,4-dimethyl-morpholin-4...)
Affinity DataIC50:  4.00E+6nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT); Range = 1300-4000 microMMore data for this Ligand-Target Pair
In DepthDetails Article