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Found 694 with Last Name = 'bhatia' and Initial = 'pa'
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50102712(2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyraz...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145078(2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-b...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145081(2-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145081(2-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  8.70nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145076(2-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145076(2-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145084(2-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  14.8nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145084(2-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  14.8nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145072(2-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-b...)
Affinity DataKi:  20.4nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474632(CHEMBL327116)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474632(CHEMBL327116)
Affinity DataKi:  23nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145083(2-[4-(3-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-b...)
Affinity DataKi:  26.5nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  33nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  36nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  45nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474631(CHEMBL323004)
Affinity DataKi:  46nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataKi:  47nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  48nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  49nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145079(2-(4-Phenyl-piperazin-1-ylmethyl)-1H-benzoimidazol...)
Affinity DataKi:  52nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  72nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145080(2-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-be...)
Affinity DataKi:  79.6nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474642(CHEMBL110975)
Affinity DataKi:  83nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474638(CHEMBL111463)
Affinity DataKi:  85nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474637(CHEMBL2111710)
Affinity DataKi:  91nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  98nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474644(CHEMBL112814)
Affinity DataKi:  100nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  105nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  115nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of bovine clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474666(CHEMBL321644)
Affinity DataKi:  123nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474643(CHEMBL111734)
Affinity DataKi:  129nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataKi:  132nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  135nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  138nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of bovine clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(HAMSTER)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  145nMAssay Description:In vitro binding affinity towards alpha-1B adrenergic receptor of hamster clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474635(CHEMBL109827)
Affinity DataKi:  148nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of bovine clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474673(CHEMBL110751)
Affinity DataKi:  166nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145075(2-((4-(pyridin-2-yl)piperazin-1-yl)methyl)-1H-benz...)
Affinity DataKi:  167nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  170nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  186nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  191nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  195nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474638(CHEMBL111463)
Affinity DataKi:  204nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(HAMSTER)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474644(CHEMBL112814)
Affinity DataKi:  214nMAssay Description:In vitro binding affinity towards alpha-1B adrenergic receptor of hamster clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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