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Found 270 with Last Name = 'bianucci' and Initial = 'am'
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196014(3-(2-(trifluoromethyl)benzyl)-N-cyclopentyl-5-phen...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106372(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  0.710nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196002(3-(2-fluorobenzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3...)
Affinity DataKi:  1.15nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106373(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  1.40nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196009(3-benzyl-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106374(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  2.10nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276769(CHEMBL514399 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106376(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  2.30nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276770(CHEMBL456211 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195990(3-(2-fluorobenzyl)-5-phenyl-N-propyl-3H-[1,2,3]tri...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195996(3-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM106370(9-(ortho-fluorobenzyl)-2-phenyl-azaadenine (1bis))
Affinity DataKi:  3.80nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196018(3-(2-fluorobenzyl)-N-butyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195995(1-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195992(3-benzyl-N-cyclobutyl-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106378(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  5.5nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106375(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  5.5nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276243(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimid...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196015(3-(2-(trifluoromethyl)benzyl)-N-butyl-5-phenyl-3H-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196003(3-(2-fluorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196030(3-(2-(trifluoromethyl)benzyl)-N-cyclohexyl-5-pheny...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276242(4-amino-N-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195999(1-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyri...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276707(CHEMBL458346 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196020(3-(2-(trifluoromethyl)benzyl)-N-cyclopropyl-5-phen...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276772(CHEMBL456011 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196011(3-(2-chlorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106371(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  9.20nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276867(CHEMBL459772 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196010(3-(2-fluorobenzyl)-N-ethyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195997(3-(2-chlorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196012(3-benzyl-N-butyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196022(3-benzyl-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195994(3-benzyl-N-cyclopropyl-5-phenyl-3H-[1,2,3]triazolo...)
Affinity DataKi:  11.3nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276866(CHEMBL517097 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276771(CHEMBL456010 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196023(3-benzyl-N-hexyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d...)
Affinity DataKi:  13.2nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106381(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  14nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196026(3-(2-(trifluoromethyl)benzyl)-N-methyl-5-phenyl-3H...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195998(3-(2-fluorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106384(N-[9-ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6-...)
Affinity DataKi:  18nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196007(3-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyri...)
Affinity DataKi:  21.4nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276939(CHEMBL517258 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195993(3-(2-chlorobenzyl)-N-cyclobutyl-5-phenyl-3H-[1,2,3...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276161(CHEMBL471022 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196019(3-(2-fluorobenzyl)-N-methyl-5-phenyl-3H-[1,2,3]tri...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196024(3-(2-fluorobenzyl)-N-hexyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50242664(CHEMBL455383 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106380(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  28nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196016(3-(2-chlorobenzyl)-N-hexyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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