Compile Data Set for Download or QSAR
maximum 50k data
Found 53 with Last Name = 'boissard' and Initial = 'cg'
LigandPNGBDBM50038163((6,7-Dichloro-2,3-dioxo-3,4-dihydro-2H-quinoxalin-...)
Affinity DataKi:  110nMAssay Description:Binding affinity for glycine site-NMDA receptor was determined by the ability to displace [3H]glycine in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281275((6,7-Dimethyl-2,3-dioxo-3,4-dihydro-2H-quinoxalin-...)
Affinity DataKi:  5.28E+3nMAssay Description:Binding affinity for glycine site-NMDA receptor was determined by the ability to displace [3H]glycine in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281273((6,7-Dimethyl-2,3-dioxo-3,4-dihydro-2H-quinoxalin-...)
Affinity DataKi:  1.38E+4nMAssay Description:Binding affinity for glycine site-NMDA receptor was determined by the ability to displace [3H]glycine in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171275((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition against Cytochrome P450 2C9 prepared from baculovirus-infected insect cells using 7-methoxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171277(CHEMBL195561 | [4-(5-Chloro-2-hydroxy-phenyl)-3-(2...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition against Cytochrome P450 2C9 prepared from baculovirus-infected insect cells using 7-methoxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition against Cytochrome P450 2C19 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171284(4-(5-Chloro-2-methoxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50:  5.47E+3nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using 7-benzyloxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171282(2-[4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethy...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition against Cytochrome P450 2C19 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171280(4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition against Cytochrome P450 2C19 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171278(12-Chloro-2-trifluoromethyl-5,7-dihydro-9-oxa-5-az...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171277(CHEMBL195561 | [4-(5-Chloro-2-hydroxy-phenyl)-3-(2...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using 7-benzyloxy- 4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171280(4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using resorufin benzyl etherMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171282(2-[4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition against Cytochrome P450 2C9 prepared from baculovirus-infected insect cells using 7-methoxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171277(CHEMBL195561 | [4-(5-Chloro-2-hydroxy-phenyl)-3-(2...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using resorufin benzyl etherMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171280(4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition against Cytochrome P450 2C9 prepared from baculovirus-infected insect cells using 7-methoxy-4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171283(2-Chloro-6-(2-oxo-propyl)-11-trifluoromethyl-6,8-d...)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171277(CHEMBL195561 | [4-(5-Chloro-2-hydroxy-phenyl)-3-(2...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition against Cytochrome P450 2D6 prepared from baculovirus-infected insect cells using 3-[2-(N,N-diethyl-N-methylamino)ethyl]-7- methoxy-4-meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171277(CHEMBL195561 | [4-(5-Chloro-2-hydroxy-phenyl)-3-(2...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition against Cytochrome P450 2C19 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171282(2-[4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethy...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using 7-benzyloxy- 4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171280(4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using 7-benzyloxy- 4-trifluoromethylcoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition against Cytochrome P450 1A2 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition against Cytochrome P450 2D6 prepared from baculovirus-infected insect cells using 3-[2-(N,N-diethyl-N-methylamino)ethyl]-7-methoxy-4-methy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171279(4-(5-Chloro-2-hydroxy-phenyl)-3-[3-((S)-diethyl-am...)
Affinity DataIC50:  3.77E+4nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171277(CHEMBL195561 | [4-(5-Chloro-2-hydroxy-phenyl)-3-(2...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition against Cytochrome P450 1A2 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171282(2-[4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethy...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using resorufin benzyl etherMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171276(4-(5-Chloro-2-hydroxy-phenyl)-3-[3-((R)-diethyl-am...)
Affinity DataIC50:  5.07E+4nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171282(2-[4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition against Cytochrome P450 1A2 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50241125((+)-4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition against Cytochrome P450 3A4 prepared from baculovirus-infected insect cells using resorufin benzyletherMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171280(4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition against Cytochrome P450 1A2 prepared from baculovirus-infected insect cells using 3-cyano-7-ethoxycoumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171281(1-(4-Benzyl-2-oxo-1,2-dihydro-quinolin-3-yl)-pyrid...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171282(2-[4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition against Cytochrome P450 2D6 prepared from baculovirus-infected insect cells using 3-[2-(N,N-diethyl-N-methylamino)ethyl]-7- methoxy-4-meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50171280(4-(5-Chloro-2-hydroxy-phenyl)-3-(2-hydroxy-ethyl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition against Cytochrome P450 2D6 prepared from baculovirus-infected insect cells using 3-[2-(N,N-diethyl-N-methylamino)ethyl]-7- methoxy-4-meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50442470(CHEMBL401942)
Affinity DataEC50:  2.40nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50410081(CHEMBL361184)
Affinity DataEC50:  10nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50410077(CHEMBL180886)
Affinity DataEC50:  20nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143560((E)-N-[(S)-1-(4-Cyclopropylmethyl-3,4-dihydro-2H-b...)
Affinity DataEC50:  60nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)
Affinity DataEC50:  1.30E+3nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50130610((E)-N-[(S)-1-(3-Morpholin-4-yl-phenyl)-ethyl]-3-ph...)
Affinity DataEC50:  3.20E+3nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50442469(CHEMBL2440362)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50442468(CHEMBL2440364)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of mouse KCNQ2 expressed in HEK293 cells at -40 mV holding potential by whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50142346(CHEMBL41078 | N-[4-(5-Chloro-2-hydroxy-benzyl)-2-o...)
Affinity DataEC50:  663nMAssay Description:Increased outward current at -40 mV mediated by mouse KCNQ2 channel expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143561((E)-N-[(S)-1-(3,4-Dihydro-2H-benzo[1,4]oxazin-6-yl...)
Affinity DataEC50:  2.00E+3nMAssay Description:Whole-cell patch-clamp on recombinant mouse KCNQ2 channels expressed in HEK 293 cells at -40 mVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143559((E)-N-[1-((S)-4-Ethyl-3,4-dihydro-2H-benzo[1,4]oxa...)
Affinity DataEC50:  200nMAssay Description:Whole-cell patch-clamp on recombinant mouse KCNQ2 channels expressed in HEK 293 cells at -40 mVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143560((E)-N-[(S)-1-(4-Cyclopropylmethyl-3,4-dihydro-2H-b...)
Affinity DataEC50:  60nMAssay Description:Whole-cell patch-clamp on recombinant mouse KCNQ2 channels expressed in HEK 293 cells at -40 mVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)
Affinity DataEC50:  1.30E+3nMAssay Description:Whole-cell patch-clamp on recombinant mouse KCNQ2 channels expressed in HEK 293 cells at -40 mVMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50130610((E)-N-[(S)-1-(3-Morpholin-4-yl-phenyl)-ethyl]-3-ph...)
Affinity DataEC50:  3.28E+3nMAssay Description:Whole-cell patch-clamp on recombinant mouse KCNQ2 channels expressed in HEK 293 cells at -40 mVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Mus musculus)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50143557((E)-3-(2-Fluoro-phenyl)-N-[1-((S)-4-methyl-3,4-dih...)
Affinity DataEC50:  940nMAssay Description:Whole-cell patch-clamp on recombinant mouse KCNQ2 channels expressed in HEK 293 cells at -40 mVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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