Affinity DataKi: 0.0500nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Binding affinity against HIV-1 aspartic proteinase was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: <1nMAssay Description:Binding affinity against HIV-1 aspartic proteinase was determinedMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity against HIV-1 aspartic proteinase was determinedMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 118nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 437nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 780nMAssay Description:Binding affinity against HIV-1 aspartic proteinase was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+3nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 3.13E+3nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Harvard University
Curated by ChEMBL
Harvard University
Curated by ChEMBL
Affinity DataKi: 6.50E+3nMAssay Description:Binding affinity towards human immunodeficiency virus type 1 protease determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 8.10E+3nMAssay Description:Predicted binding affinity for beta secretase by linear interaction energy continuum electrostaticsMore data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nMAssay Description:Predicted binding affinity for beta secretase by linear interaction energy continuum electrostaticsMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+3nMAssay Description:Predicted binding affinity for beta secretase by linear interaction energy continuum electrostaticsMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+4nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of Helicobacter pylori DHQ2More data for this Ligand-Target Pair
Affinity DataKi: 2.24E+4nMAssay Description:Binding affinity towards Beta-secretase determined using continuum electrostatics solvationMore data for this Ligand-Target Pair