TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono...More data for this Ligand-Target Pair
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged bacterial Escherichia coli TEM-1 (24 to 286 residues) expressed in Escherichia coli BL21 (DE3) cells ...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 3.24E+4nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 3.24E+4nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
Affinity DataIC50: 3.28E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged bacterial Escherichia coli TEM-1 (24 to 286 residues) expressed in Escherichia coli BL21 (DE3) cells ...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
University Of Turin
Curated by ChEMBL
University Of Turin
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant N-terminal His6-tagged DHODH (159-569 residues) expressed in Escherichia coli BL21(DE3) using DHO as ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of C-terminal His10-tagged Escherichia coli B ER2560 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leuco...More data for this Ligand-Target Pair
Affinity DataIC50: 3.73E+4nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa OXA-10 expressed in Escherichia coli BL21 (DE3) cells using FC5 as substrate preincubated up to 360 ...More data for this Ligand-Target Pair
TargetAcyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase(Escherichia coli (Enterobacteria))
X-Biotix Therapeutics
Curated by ChEMBL
X-Biotix Therapeutics
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant Escherichia coli LpxA using UDP-GlcNAc as substrate incubated for 30 mins by spectrophotometric methodMore data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 5.27E+4nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
University Of Warwick
Curated by ChEMBL
University Of Warwick
Curated by ChEMBL
Affinity DataIC50: 5.27E+4nMAssay Description:Inhibition of C-terminal His10-tagged Staphylococcus aureus seg50 SerRS expressed in Lemo21(DE3) using Ap4A as substrate in presence of serine by leu...More data for this Ligand-Target Pair
Affinity DataIC50: 6.73E+4nMAssay Description:Inhibition of human N-terminal polyHis-tagged SerRS expressed in Escherichia coli BL21 (DE3) using Ap4A as substrate in presence of serine by leucono...More data for this Ligand-Target Pair