Affinity DataKi: 0.110nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Antagonist activity at mouse wild type 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF as...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Inhibitory activity against Monoamine oxidase BMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Non-selective inhibitory activity was determined against 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 7 receptor was determined in HEK293 cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards human recombinant 5-hydroxytryptamine 7 receptor was determined using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards human recombinant 5-hydroxytryptamine 7 receptor was determined using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 7 receptor was determined in HEK293 cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]-GR-113,808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneChecked by AuthorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Universitat AutòNoma De Barcelona
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibitory activity against Monoamine oxidase BMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 7 receptor was determined in HEK293 cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity towards human recombinant 5-hydroxytryptamine 7 receptor was determined using [3H]5-CT as radioligandMore data for this Ligand-Target Pair