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Found 145 with Last Name = 'canning' and Initial = 'p'
TargetDiscoidin domain-containing receptor 2(Homo sapiens (Human))
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM50237710(4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...)
Affinity DataIC50:  0.5nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056508(CHEMBL3341945)
Affinity DataIC50:  4nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056507(CHEMBL3341944)
Affinity DataIC50:  6nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056506(CHEMBL3341943 | US10688093, Compound 382_0087_6488...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613268(CHEMBL5275681)
Affinity DataIC50:  9nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056680(CHEMBL3341794)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056508(CHEMBL3341945)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613266(CHEMBL5268562)
Affinity DataIC50:  11nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613282(CHEMBL5270264)
Affinity DataIC50:  13nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056510(CHEMBL3341947)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056675(CHEMBL3341787)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056508(CHEMBL3341945)
Affinity DataIC50:  16nMAssay Description:Inhibition of BMP2-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056507(CHEMBL3341944)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056684(CHEMBL3341941 | US10688093, Compound 382_0087_7249...)
Affinity DataIC50:  20nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056680(CHEMBL3341794)
Affinity DataIC50:  20nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056509(CHEMBL3341946)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056676(CHEMBL3341789)
Affinity DataIC50:  24nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056676(CHEMBL3341789)
Affinity DataIC50:  27nMAssay Description:Inhibition of ALK1 (unknown origin) expressed in HEK293T cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056676(CHEMBL3341789)
Affinity DataIC50:  27nMAssay Description:Inhibition of ALK2 (unknown origin) expressed in HEK293T cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613267(CHEMBL5276443)
Affinity DataIC50:  27nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056508(CHEMBL3341945)
Affinity DataIC50:  27nMAssay Description:Inhibition of BMP4-induced BMP receptor in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056680(CHEMBL3341794)
Affinity DataIC50:  30nMAssay Description:Inhibition of purified human ALK5 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056675(CHEMBL3341787)
Affinity DataIC50:  30nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM102619(K02288a | US10688093, Compound 382_0087_0284 | US1...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613281(CHEMBL5270195)
Affinity DataIC50:  36nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613279(CHEMBL5290255)
Affinity DataIC50:  37nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613283(CHEMBL5271729)
Affinity DataIC50:  38nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613280(CHEMBL5276347)
Affinity DataIC50:  39nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056510(CHEMBL3341947)
Affinity DataIC50:  40nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM50237710(4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...)
Affinity DataIC50:  43nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104010(DDR1-IN-2)
Affinity DataIC50:  47.6nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056507(CHEMBL3341944)
Affinity DataIC50:  49nMAssay Description:Inhibition of purified human ALK5 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613269(CHEMBL5291180)
Affinity DataIC50:  50nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056506(CHEMBL3341943 | US10688093, Compound 382_0087_6488...)
Affinity DataIC50:  60nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056549(CHEMBL3341952)
Affinity DataIC50:  63nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056511(CHEMBL3341948)
Affinity DataIC50:  86nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056685(CHEMBL3341942)
Affinity DataIC50:  90nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613284(CHEMBL5269867)
Affinity DataIC50:  96nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056676(CHEMBL3341789)
Affinity DataIC50:  100nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056508(CHEMBL3341945)
Affinity DataIC50:  100nMAssay Description:Inhibition of TGFbeta1-induced TGFbeta type 1 ALK5 in HEK293T cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104009(DDR1-IN-1)
Affinity DataIC50:  105nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056678(CHEMBL3341792)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056674(CHEMBL3341953)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056511(CHEMBL3341948)
Affinity DataIC50:  110nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM225684(GTC000457A)
Affinity DataIC50:  110nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056507(CHEMBL3341944)
Affinity DataIC50:  110nMAssay Description:Inhibition of TGFbeta1-induced TGFbeta type 1 ALK5 in HEK293T cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1(Homo sapiens (Human))
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056677(CHEMBL3341791)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant human ALK2 kinase after 45 mins by liquid scintillation counting in presence of ATP [gamma-32P]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613285(CHEMBL5277663)
Affinity DataIC50:  120nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50613270(CHEMBL5288117)
Affinity DataIC50:  130nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetActivin receptor type-1(Mus musculus)
Massachusetts Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50056509(CHEMBL3341946)
Affinity DataIC50:  140nMAssay Description:Inhibition of BMP6-induced BMP receptor type 1 ALK2 in mouse C2C12 cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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