Compile Data Set for Download or QSAR
maximum 50k data
Found 61 with Last Name = 'casebier' and Initial = 'd'
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378919(CHEMBL2011218)
Affinity DataIC50:  0.0400nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378913(CHEMBL2011227)
Affinity DataIC50:  0.0500nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378927(CHEMBL2011226)
Affinity DataIC50:  0.0500nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378917(CHEMBL2011216)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378916(CHEMBL2011215)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378925(CHEMBL2011224)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378914(CHEMBL2011213)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378935(CHEMBL2011235)
Affinity DataIC50:  0.140nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378915(CHEMBL2011214)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378918(CHEMBL2011217)
Affinity DataIC50:  0.25nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378926(CHEMBL2011225)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378928(CHEMBL2011228)
Affinity DataIC50:  0.350nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378923(CHEMBL2011222)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378920(CHEMBL2011219)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378922(CHEMBL2011221)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378924(CHEMBL2011223)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378934(CHEMBL2011234)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378936(CHEMBL2011236)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378930(CHEMBL2011230)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378933(CHEMBL2011233)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378932(CHEMBL2011232)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378921(CHEMBL2011220)
Affinity DataIC50:  21nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378929(CHEMBL2011229)
Affinity DataIC50:  26nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378931(CHEMBL2011231)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H](-)-CGP-12177 from adrenergic beta1 receptor by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28928((2S,3S)-N-(3-chlorophenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  1.83E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28929((2S,3S)-N-(2-chlorophenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  5.66E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28930((2S,3S)-N-(4-fluorophenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  4.24E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28921((2S,3S)-N-(4-bromophenyl)-1-hydroxy-3-methylpentan...)
Affinity DataEC50:  2.21E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28931((2S,3S)-N-(4-cyanophenyl)-1-hydroxy-3-methylpentan...)
Affinity DataEC50: >1.00E+5nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28932((2S,3S)-1-hydroxy-3-methyl-N-(4-methylphenyl)penta...)
Affinity DataEC50:  1.43E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28933((2S,3S)-1-hydroxy-3-methyl-N-[4-(trifluoromethyl)p...)
Affinity DataEC50:  1.31E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28934((2S,3S)-N-(4-acetylphenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  6.02E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28935((2S,3S)-1-hydroxy-N-(4-methanesulfonylphenyl)-3-me...)
Affinity DataEC50: >1.00E+5nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28936((2S,3S)-1-hydroxy-3-methyl-N-(4-nitrophenyl)pentan...)
Affinity DataEC50:  2.09E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM28937((2S,3S)-N-[4-(1,1-difluoroethoxy)phenyl]-1-hydroxy...)
Affinity DataEC50:  2.35E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM28938((2S,3S)-N-(3,4-dichlorophenyl)-1-hydroxy-3-methylp...)
Affinity DataEC50:  3.70E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28920((2S,3S)-N-(4-chlorophenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  5.45E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28961(CHEMBL180641 | ethyl 4-[(4-chlorobenzene)sulfonyl]...)
Affinity DataEC50:  1.22E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28960((2R)-2-{[5-chloro-2-(hydroxymethyl)phenyl](4-chlor...)
Affinity DataEC50:  85nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28959((3S,4S)-N-(4-chlorophenyl)-2-hydroxy-2,4-dimethylh...)
Affinity DataEC50: >1.00E+5nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28958((3S,4S)-N-(4-chlorophenyl)-2-hydroxy-4-methylhexan...)
Affinity DataEC50:  4.93E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28957((1S)-N-(4-chlorophenyl)-2-hydroxy-1-phenylethane-1...)
Affinity DataEC50:  6.88E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28956((1S)-N-(4-chlorophenyl)-1-cyclohexyl-2-hydroxyetha...)
Affinity DataEC50:  1.12E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28955((2S,3R)-N-(4-chlorophenyl)-1-hydroxy-3-methylpenta...)
Affinity DataEC50:  758nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28954((2S)-N-(4-chlorophenyl)-1-hydroxy-4-methylpentane-...)
Affinity DataEC50:  1.53E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28923((2S)-N-(4-chlorophenyl)-3-ethyl-1-hydroxypentane-2...)
Affinity DataEC50:  294nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28953((2S)-N-(4-chlorophenyl)-1-hydroxy-3,3-dimethylbuta...)
Affinity DataEC50:  2.91E+4nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28952((2S)-N-(4-chlorophenyl)-1-hydroxy-3-methylbutane-2...)
Affinity DataEC50:  4.58E+3nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28951((2S)-N-(4-chlorophenyl)-1-hydroxybutane-2-sulfonam...)
Affinity DataEC50: >1.00E+5nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28950((2S)-N-(4-chlorophenyl)-1-hydroxypropane-2-sulfona...)
Affinity DataEC50: >1.00E+5nMAssay Description:A Chinese Hamster Ovary cell line stably expressing human beta-APP were aliquoted into a 96-well plate, and after attachment the medium was replaced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 61 total ) | Next | Last >>
Jump to: