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Found 88 with Last Name = 'castellano' and Initial = 'r'
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50:  20nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50:  71nMAssay Description:Inhibition of BRD2-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586230(CHEMBL5081350)
Affinity DataIC50:  72nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50:  72nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  85nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50:  98nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586228(CHEMBL5077541)
Affinity DataIC50:  100nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  120nMAssay Description:Inhibition of BRD2-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50:  130nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586226(CHEMBL5069987)
Affinity DataIC50:  140nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586236(CHEMBL5083228)
Affinity DataIC50:  150nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586243(CHEMBL5072385)
Affinity DataIC50:  170nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586242(CHEMBL5074953)
Affinity DataIC50:  170nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586238(CHEMBL5089658)
Affinity DataIC50:  210nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586239(CHEMBL5094390)
Affinity DataIC50:  210nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586233(CHEMBL5077199)
Affinity DataIC50:  220nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586227(CHEMBL5079297)
Affinity DataIC50:  300nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586244(CHEMBL5086321)
Affinity DataIC50:  320nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  325nMAssay Description:Binding affinity to human partial length BRD3-BD2 (G306 to P416) expressed in bacterial system assessed as dissociation constant by BROMOscan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586237(CHEMBL5075819)
Affinity DataIC50:  380nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586240(CHEMBL5076502)
Affinity DataIC50:  410nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586224(CHEMBL5085041)
Affinity DataIC50:  410nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586232(CHEMBL5089846)
Affinity DataIC50:  420nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586229(CHEMBL5089257)
Affinity DataIC50:  440nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586247(CHEMBL5075514)
Affinity DataIC50:  470nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586235(CHEMBL5094939)
Affinity DataIC50:  490nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586241(CHEMBL5090901)
Affinity DataIC50:  530nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586231(CHEMBL5090190)
Affinity DataIC50:  570nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586234(CHEMBL5081830)
Affinity DataIC50:  630nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586246(CHEMBL5074555)
Affinity DataIC50:  740nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  775nMAssay Description:Binding affinity to human partial length BRD4-BD2 (K333 to E460 residues) expressed in bacterial system assessed as dissociation constant by BROMOsca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586219(CHEMBL5077591)
Affinity DataIC50:  800nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586245(CHEMBL5076250)
Affinity DataIC50:  880nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586216(CHEMBL5078986)
Affinity DataIC50:  900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586220(CHEMBL5084945)
Affinity DataIC50:  900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586221(CHEMBL5075052)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586217(CHEMBL5084236)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586245(CHEMBL5076250)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586244(CHEMBL5086321)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586218(CHEMBL5093626)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586231(CHEMBL5090190)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586229(CHEMBL5089257)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  2.60E+3nMAssay Description:Binding affinity to human partial length BRD2-BD2 (E348 to D455) expressed in bacterial system assessed as dissociation constant by BROMOscan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586228(CHEMBL5077541)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586233(CHEMBL5077199)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586235(CHEMBL5094939)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586221(CHEMBL5075052)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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