Affinity DataKi: 0.00780nMAssay Description:Binding affinity to human BK1 receptor E273 mutantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0340nMAssay Description:Binding affinity to human BK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0380nMAssay Description:Binding affinity to human BK1 receptor N298 mutantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0450nMAssay Description:Binding affinity to human BK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0490nMAssay Description:Binding affinity to human BK1 receptor D291 mutantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity to human BK1 receptor E273 mutantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to human BK1 receptor D291 mutantMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Affinity DataKi: 0.350nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]des-arg10leu9kallidin from human bradykinin B1 receptor expressed in CHO cells by Wallac beta-plate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]-SCH-23,390 from rat striatal ...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]des-arg10leu9kallidin from human bradykinin B1 receptor expressed in CHO cells by Wallac beta-plate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity to human BK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity of compound evaluated for Opioid receptor mu 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity to human BK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity of compound evaluated for Opioid receptor mu 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]des-arg10leu9kallidin from human bradykinin B1 receptor expressed in CHO cells by Wallac beta-plate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]des-arg10leu9kallidin from human bradykinin B1 receptor expressed in CHO cells by Wallac beta-plate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair