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Found 11 with Last Name = 'chapuis' and Initial = 'jc'
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292348(CHEMBL501262 | bryostatin 10)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292349(CHEMBL505767 | bryostatin 18)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292351(CHEMBL509516 | bryostatin 16)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50292350(CHEMBL452391 | bryostatin 17 | delta 19,20-bryosta...)
Affinity DataKi:  188nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM23940(1,3-dimethoxy-5-[(Z)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of tubulin polymerization reported as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of tubulin polymerization reported as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50473760(3,4'',5-Trismethoxybenzophenone | CHEMBL86124)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of tubulin polymerization reported as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50156812(PHENSTATIN)
Affinity DataIC50:  3.45E+3nMAssay Description:Inhibition of tubulin polymerization reported as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50069241(CHEMBL405162 | Spongistatin-1)
Affinity DataIC50:  3.60E+3nMAssay Description:Compound was tested for its ability to inhibit the glutamate induced polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50473759(CHEMBL87712)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of tubulin polymerization reported as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerization reported as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed