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Found 78 with Last Name = 'chen' and Initial = 'hz'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092959(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.110nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092961(1-(isopropylsulfonyl)-4-(4-(1-(4-(4-methoxyphenyls...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092969(CHEMBL74117 | Cyclopropyl-(4-{1-[4-(4-methoxy-benz...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092958(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)p...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092962(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092968(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.350nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092974(1'-Benzenesulfonyl-4-{1-[4-(4-methoxy-benzenesulfo...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092960(1'-(Butane-1-sulfonyl)-4-{1-[4-(4-methoxy-benzenes...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092965(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092973(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092963(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092970(1'-Ethanesulfonyl-4-{1-[4-(4-methoxy-benzenesulfon...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092972(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092964(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  0.991nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092957(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)-1-(...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092966(1-(benzylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulf...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092971(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092975(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  3nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092967(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092959(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  6.5nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092957(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)-1-(...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092968(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092962(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  10nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092963(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  11nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092973(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  15nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092958(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)p...)
Affinity DataKi:  26nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092961(1-(isopropylsulfonyl)-4-(4-(1-(4-(4-methoxyphenyls...)
Affinity DataKi:  32nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092966(1-(benzylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulf...)
Affinity DataKi:  33nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092974(1'-Benzenesulfonyl-4-{1-[4-(4-methoxy-benzenesulfo...)
Affinity DataKi:  37nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092972(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  41nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092965(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  42nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092960(1'-(Butane-1-sulfonyl)-4-{1-[4-(4-methoxy-benzenes...)
Affinity DataKi:  57nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092964(4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}...)
Affinity DataKi:  60nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092967(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  61nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092969(CHEMBL74117 | Cyclopropyl-(4-{1-[4-(4-methoxy-benz...)
Affinity DataKi:  68nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092970(1'-Ethanesulfonyl-4-{1-[4-(4-methoxy-benzenesulfon...)
Affinity DataKi:  74nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092975(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  96nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50092971(1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)viny...)
Affinity DataKi:  117nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427125(CHEMBL2323444)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427129(CHEMBL2323441)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427131(CHEMBL2323446)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427127(CHEMBL2323442)
Affinity DataKi:  3.70E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427129(CHEMBL2323441)
Affinity DataKi:  8.80E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427127(CHEMBL2323442)
Affinity DataKi:  9.80E+3nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427131(CHEMBL2323446)
Affinity DataKi:  1.07E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427125(CHEMBL2323444)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427126(CHEMBL2323443)
Affinity DataKi:  6.60E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427130(CHEMBL2323447)
Affinity DataKi:  7.10E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427130(CHEMBL2323447)
Affinity DataKi:  7.70E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50427128(CHEMBL2321893)
Affinity DataKi:  8.30E+4nMAssay Description:Displacement of [3H]NMS from muscarinic M3 receptor in Sprague-Dawley rat submandibulary gland after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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