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Found 43 with Last Name = 'chen' and Initial = 'nn'
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50005782(ATI-13387X | ONALESPIB)
Affinity DataIC50:  13nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50450705(CHEMBL4170630)
Affinity DataIC50:  20nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587115(CHEMBL5093243)
Affinity DataIC50:  60nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587119(CHEMBL5089044)
Affinity DataIC50:  100nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587134(CHEMBL5079918)
Affinity DataIC50:  203nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587116(CHEMBL5084235)
Affinity DataIC50:  205nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587120(CHEMBL5090316)
Affinity DataIC50:  210nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587132(CHEMBL5089381)
Affinity DataIC50:  234nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587118(CHEMBL5084137)
Affinity DataIC50:  251nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587130(CHEMBL5094079)
Affinity DataIC50:  310nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587114(CHEMBL5087678)
Affinity DataIC50:  313nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587113(CHEMBL5093787)
Affinity DataIC50:  325nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587133(CHEMBL5090818)
Affinity DataIC50:  393nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587117(CHEMBL5087889)
Affinity DataIC50:  519nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587138(CHEMBL5084856)
Affinity DataIC50:  528nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587137(CHEMBL5087347)
Affinity DataIC50:  627nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587139(CHEMBL5091405)
Affinity DataIC50:  797nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587112(CHEMBL5075059)
Affinity DataIC50:  914nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587131(CHEMBL5077310)
Affinity DataIC50:  947nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587142(CHEMBL5090524)
Affinity DataIC50:  985nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587140(CHEMBL5070758)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587141(CHEMBL5093202)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587135(CHEMBL5088257)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587129(CHEMBL5087473)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587145(CHEMBL5092629)
Affinity DataIC50:  2.05E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587127(CHEMBL5089184)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587144(CHEMBL5075220)
Affinity DataIC50:  2.41E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587126(CHEMBL5081112)
Affinity DataIC50:  2.77E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587128(CHEMBL5089014)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587143(CHEMBL5077569)
Affinity DataIC50:  4.78E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587123(CHEMBL5076003)
Affinity DataIC50:  6.84E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587125(CHEMBL5082207)
Affinity DataIC50:  7.54E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587124(CHEMBL5085266)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587136(CHEMBL5088079)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587121(CHEMBL5091953)
Affinity DataIC50:  6.26E+4nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587122(CHEMBL5092143)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)
Affinity DataKd: >2.50E+5nMAssay Description:Binding affinity to Hsp90alpha (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmin(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataKd:  200nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmin(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)
Affinity DataKd:  220nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmin(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587146(CHEMBL5073759)
Affinity DataKd:  200nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587115(CHEMBL5093243)
Affinity DataKon:  0.114M-1s-1Assay Description:Binding affinity to His-tagged human N-terminal HSP90alpha (1 to 236 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataKd:  8.20E+3nMAssay Description:Binding affinity to Hsp90alpha (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmin(Canis familiaris)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587115(CHEMBL5093243)
Affinity DataKon:  0.0284M-1s-1Assay Description:Binding affinity to GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant at 0.37 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed