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Found 41 with Last Name = 'chen' and Initial = 'st'
TargetChymotrypsinogen A(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50283074(CHEMBL413681 | Cyclic-Ac-Asp-Ile-Val-Thr-Met-Glu-T...)
Affinity DataKi:  191nMAssay Description:Compound was tested for the inhibition of chymotrypsin at 120 nMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsinogen A(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50283074(CHEMBL413681 | Cyclic-Ac-Asp-Ile-Val-Thr-Met-Glu-T...)
Affinity DataKi:  203nMAssay Description:Compound was tested for the inhibition of chymotrypsin at 69 nMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsinogen A(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50283075(CHEMBL269484 | Cyclic-NH2-Glu-Thr -Met-Glu-Tyr-Arg...)
Affinity DataKi:  656nMAssay Description:Compound was tested for the inhibition of chymotrypsin at 276 nMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsinogen A(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50283075(CHEMBL269484 | Cyclic-NH2-Glu-Thr -Met-Glu-Tyr-Arg...)
Affinity DataKi:  668nMAssay Description:Compound was tested for the inhibition of chymotrypsin at 138 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50044355(2,5-Dibutyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50:  5nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283548(1-{(5S,8S)-3-Butyl-1-chloro-5-[2'-(2H-tetrazol-5-y...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283551(1-{(5S,8S)-3-Butyl-5-[2'-(2H-tetrazol-5-yl)-biphen...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283562(5-[4'-(2,4-Dibutyl-imidazol-1-ylmethyl)-biphenyl-2...)
Affinity DataIC50:  63nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283557(3-Butyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283564(1,3-Dibutyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50:  190nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283565(2-Butyl-5-propyl-4-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  500nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283555(2-Butyl-8-propyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283555(2-Butyl-8-propyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM35440(ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...)
Affinity DataIC50:  7.82E+3nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50283550(1-{(5S,7R,8R)-7-Bromo-3-butyl-5-[2'-(2-trityl-2H-t...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283549(2,5-Dibutyl-4-[2'-(2-trityl-2H-tetrazol-5-yl)-biph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283566(5-[1-(2-Bromo-ethyl)-butyl]-2-butyl-4-[2'-(2-trity...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283556(2-Butyl-8-propyl-5-[2'-(2-trityl-2H-tetrazol-5-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283561(1-{(5S,8S)-3-Butyl-5-[2'-(2-trityl-2H-tetrazol-5-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283560(2-Butyl-5-[1-(4,4-dimethyl-4,5-dihydro-oxazol-2-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283559(8-Propyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283558(2-Butyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283563(2-Butyl-5-[1-(2-hydroxy-ethyl)-butyl]-4-[2'-(2-tri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283553(5-[4'-(2,4-Dibutyl-imidazol-1-ylmethyl)-biphenyl-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283554(5-(1-Bromo-butyl)-2-butyl-4-[2'-(2-trityl-2H-tetra...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283556(2-Butyl-8-propyl-5-[2'-(2-trityl-2H-tetrazol-5-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283557(3-Butyl-5-[2'-(2H-tetrazol-5-yl)-biphenyl-4-yl]-5,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208873(2-chloro-6(methylamino)purine | CHEMBL446449)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM33218(Adenine, 1 | CHEMBL226345 | purine, 6)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208876(1H-Pyrazolo[3,4-d]pyrimidin-4-ylamine | 4-aminopyr...)
Affinity DataIC50:  3.03E+4nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50283552(2-Butyl-5-propyl-4-[1-[2'-(2H-tetrazol-5-yl)-biphe...)
Affinity DataIC50:  4.50E+4nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208881(5-Nitro-1H-benzoimidazole | 5-nitrobenzimidazole |...)
Affinity DataIC50:  8.68E+4nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50200099(2-Amino-1,7-dihydro-purine-6-thione | 2-Amino-1,9-...)
Affinity DataIC50:  9.24E+4nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208872(5,6-dimethyl-1H-benzimidazole | 5,6-dimethylbenzim...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208879(2,6-diaminopurine | 9H-Purine-2,6-diamine0.5M H2SO...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208880(5-methyl-1H-benzimidazole | CHEMBL157729)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM5470(6-methoxy-9H-purin-2-amine | CHEMBL226395 | O6-Sub...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208875(2-aminopurine | 9H-Purin-2-ylamine | 9H-purin-2-am...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Biological Chemistry And The Genomics Research Center

Curated by ChEMBL
LigandPNGBDBM50208877(2-amino-6-chloropurine | 6-Cl-purine (1) | 6-chlor...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed