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Found 42 with Last Name = 'chong' and Initial = 'wk'
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM10884((2S,4S)-4-(ethylamino)-2-methyl-1,1-dioxo-2H,3H,4H...)
Affinity DataKi:  9nMAssay Description:Inhibition of human carbonic anhydrase 2 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303032(CHEMBL584939 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  13nMAssay Description:Inhibition of human carbonic anhydrase 2 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303030(6-Nitrooxy-hexanoic acid ethyl-((4S,6S)-6-methyl-7...)
Affinity DataKi:  14nMAssay Description:Inhibition of human carbonic anhydrase 2 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM10884((2S,4S)-4-(ethylamino)-2-methyl-1,1-dioxo-2H,3H,4H...)
Affinity DataKi:  43nMAssay Description:Inhibition of human carbonic anhydrase 4 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303031(CHEMBL570894 | N-Ethyl-N-((4S,6S)-6-methyl-7,7-dio...)
Affinity DataKi:  46nMAssay Description:Inhibition of human carbonic anhydrase 4 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303034(CHEMBL571337 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  63nMAssay Description:Inhibition of human carbonic anhydrase 2 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303031(CHEMBL570894 | N-Ethyl-N-((4S,6S)-6-methyl-7,7-dio...)
Affinity DataKi:  71nMAssay Description:Inhibition of human carbonic anhydrase 2 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303033(CHEMBL585756 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  76nMAssay Description:Inhibition of human carbonic anhydrase 2 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303032(CHEMBL584939 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  181nMAssay Description:Inhibition of human carbonic anhydrase 4 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303033(CHEMBL585756 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  339nMAssay Description:Inhibition of human carbonic anhydrase 4 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303032(CHEMBL584939 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  410nMAssay Description:Inhibition of human carbonic anhydrase 1 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303031(CHEMBL570894 | N-Ethyl-N-((4S,6S)-6-methyl-7,7-dio...)
Affinity DataKi:  470nMAssay Description:Inhibition of human carbonic anhydrase 1 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303033(CHEMBL585756 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  705nMAssay Description:Inhibition of human carbonic anhydrase 1 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303034(CHEMBL571337 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  1.52E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303030(6-Nitrooxy-hexanoic acid ethyl-((4S,6S)-6-methyl-7...)
Affinity DataKi:  2.95E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303034(CHEMBL571337 | Ethyl-((4S,6S)-6-methyl-7,7-dioxo-2...)
Affinity DataKi:  3.91E+3nMAssay Description:Inhibition of human carbonic anhydrase 4 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM50303030(6-Nitrooxy-hexanoic acid ethyl-((4S,6S)-6-methyl-7...)
Affinity DataKi:  4.36E+3nMAssay Description:Inhibition of human carbonic anhydrase 4 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Nicox Research Institute

Curated by ChEMBL
LigandPNGBDBM10884((2S,4S)-4-(ethylamino)-2-methyl-1,1-dioxo-2H,3H,4H...)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 by CO2 hydrase stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228277(CHEMBL1627386)
Affinity DataEC50:  2.10E+5nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50187243(17-ethinyl-3,17-estradiol | 17-ethinyl-3,17-oestra...)
Affinity DataEC50:  1.34E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228277(CHEMBL1627386)
Affinity DataEC50:  3.86E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228277(CHEMBL1627386)
Affinity DataEC50:  7.03E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50187243(17-ethinyl-3,17-estradiol | 17-ethinyl-3,17-oestra...)
Affinity DataEC50:  3.37E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228276(CHEMBL1627365)
Affinity DataEC50:  2.98E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228273(CHEMBL1627375)
Affinity DataEC50:  1.92E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228273(CHEMBL1627375)
Affinity DataEC50:  1.15E+5nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228275(CHEMBL1627370)
Affinity DataEC50:  5.12E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228275(CHEMBL1627370)
Affinity DataEC50:  4.80E+5nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228274(CHEMBL1627389)
Affinity DataEC50:  1.86E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  917nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  2.56E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228277(CHEMBL1627386)
Affinity DataEC50:  2.81E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50187243(17-ethinyl-3,17-estradiol | 17-ethinyl-3,17-oestra...)
Affinity DataEC50: >3.37E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228276(CHEMBL1627365)
Affinity DataEC50:  5.58E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228275(CHEMBL1627370)
Affinity DataEC50:  2.56E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228275(CHEMBL1627370)
Affinity DataEC50:  1.66E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228273(CHEMBL1627375)
Affinity DataEC50:  1.66E+5nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM50228274(CHEMBL1627389)
Affinity DataEC50:  7.32E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  1.83E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Sri International

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  1.83E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228273(CHEMBL1627375)
Affinity DataEC50:  5.76E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(RAT)
Sri International

Curated by ChEMBL
LigandPNGBDBM50187243(17-ethinyl-3,17-estradiol | 17-ethinyl-3,17-oestra...)
Affinity DataEC50:  1.68E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed