Compile Data Set for Download or QSAR
maximum 50k data
Found 144 with Last Name = 'christophersen' and Initial = 'p'
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50092131(1,7-diazonia-15,21-diazapentacyclo[20.6.2.27,14.08...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50061977(17,25-diazonia-2,9-diazaheptacyclo[23.6.2.24,7.210...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50048403(1,1'-(Deca-4,6-diyne-1,10-diyl)bis(4-amino-2-methy...)
Affinity DataKi:  140nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50199404(1-(3,4-Dimethoxy-benzyl)-6,7-dimethoxy-2,2-dimethy...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50377980(CHEMBL558625)
Affinity DataKi:  4.40E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM92478(Atracurium besylate | CHEMBL1360)
Affinity DataKi:  5.90E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
Affinity DataKi:  9.20E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50377979(PENUCURONIUM)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50263331((1H-Benzoimidazol-2-yl)-(R)-1,2,3,4-tetrahydronaph...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50275183(1-ethyl-1H-benzo[d]imidazol-2(3H)-one | CHEMBL4528...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50275184(6,7-dichloro-3-(hydroxyimino)indolin-2-one | CHEMB...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50275157(CHEMBL453730 | N-cyclohexyl-2-(3,5-dimethyl-1H-pyr...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM648581((1R,2S)-N1-(1-(4-fluoro-3-(trifluoromethyl)phenyl)...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648579(Methyl (S)-(1-(4-fluoro-3-(trifluoromethyl)phenyl)...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648504(US20240034717, Example 31.4 | methyl N-{[(2S)-pyrr...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648505(US20240034717, Example 31.5 | methyl N-{[(2R)-pyrr...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648506(US20240034717, Example 31.6 | methyl N-(2-amino-2-...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648507(N1-[1-(3-chlorophenyl)cyclobutyl]-2-methylpropane-...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648508(Methyl N-[1-(3-chlorophenyl)cyclobutyl]-N-{[(2S)-p...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648509(Methyl N-[1-(3-chlorophenyl)cyclobutyl]-N-{[(2R)-p...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648512(Methyl N-{[(2S)-pyrrolidin-2-yl]methyl}-N-{1-[3-(t...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648513(Methyl N-{[(2R)-pyrrolidin-2-yl]methyl}-N-{1-[3-(t...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648514(Methyl N-(2-amino-2-methylpropyl)-N-{1-[3-(trifluo...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648515(1-[4-fluoro-3-(trifluoromethyl)phenyl]-N-{[(2S)-py...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648517(N1-{1-[4-fluoro-3-(trifluoromethyl)phenyl]cyclobut...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648518(US20240034717, Example 31.18 | methyl N-{1-[4-fluo...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648519(US20240034717, Example 31.19 | methyl N-{1-[4-fluo...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648520(US20240034717, Example 31.20 | methyl N-(2-amino-2...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648522(Methyl N-{1-[3-fluoro-5-(trifluoromethyl)phenyl]cy...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648523(Methyl N-{1-[3-fluoro-5-(trifluoromethyl)phenyl]cy...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648524(Methyl N-(2-amino-2-methylpropyl)-N-{1-[3-fluoro-5...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM50547897(CHEMBL4749039 | US20240034717, Example 31.31)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM648532(Methyl ((1-aminocyclopropyl)methyl)(1-(4-fluoro-3-...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648533(Methyl 3-((1-(4-fluoro-3-(trifluoromethyl) phenyl)...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648535(N-(cyclopropylmethyl)-N-(1-(4-fluoro-3-(trifluorom...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM50547898(CHEMBL4788143 | US20240034717, Example 31.37)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50547899(CHEMBL4764429 | US20240034717, Example 31.39)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM648540(Methyl (2-amino-2-methylpropyl)(1-(3,5-dichlorophe...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648543(1-((azetidin-2-ylmethyl)(1-(4-fluoro-3-(trifluorom...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648544(Methyl (2-amino-2-methylpropyl)(1-(3-(trifluoromet...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM50547900(CHEMBL4756080 | US20240034717, Example 31.47)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50547901(CHEMBL4745327 | US20240034717, Example 31.48)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50547902(CHEMBL4785936 | US20240034717, Example 31.49)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50547903(CHEMBL4780941 | US20240034717, Example 31.50)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM648551(Methyl (R)-(1-(4-fluoro-3-(trifluoromethyl)phenyl)...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648552(Methyl (S)-(1-(4-fluoro-3-(trifluoromethyl)phenyl)...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648554(N1-(1-(4-fluoro-3-(trifluoromethyl)phenyl) cyclopr...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648555(Methyl (azetidin-2-ylmethyl)(1-(4-fluoro-3-(triflu...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM648556(Methyl (S)-(1-(4-fluoro-3-(trifluoro methyl) pheny...)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
LigandPNGBDBM50547904(CHEMBL4791725 | US20240034717, Example 31.57)
Affinity DataIC50: <300nMAssay Description:Human blood was drawn from healthy human volunteers in a standard heparinized blood sampling vial (Vacutainer, Li/heparin, ED Bioscience, Plymouth, U...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 144 total ) | Next | Last >>
Jump to: