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Found 143 with Last Name = 'cook' and Initial = 'gm'
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459080(CHEMBL4211423)
Affinity DataKi:  21nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459060(CHEMBL4208530)
Affinity DataKi:  41nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459079(CHEMBL4206764)
Affinity DataKi:  42nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459072(CHEMBL4215861)
Affinity DataKi:  42nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459071(CHEMBL4204195)
Affinity DataKi:  43nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)
Affinity DataKi:  53nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]-Ketanserin from human 5HT2A receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)
Affinity DataKi:  88nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459068(CHEMBL4212068)
Affinity DataKi:  108nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459053(CHEMBL4208241)
Affinity DataKi:  156nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459078(CHEMBL4216516)
Affinity DataKi:  166nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)
Affinity DataKi:  183nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529264(CHEMBL4513418)
Affinity DataKi:  204nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565002(CHEMBL4778666)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459073(CHEMBL4203654)
Affinity DataKi:  228nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529261(CHEMBL4445592)
Affinity DataKi:  287nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529246(CHEMBL4473654)
Affinity DataKi:  302nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459070(CHEMBL4216389)
Affinity DataKi:  315nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529247(CHEMBL4550786)
Affinity DataKi:  350nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565002(CHEMBL4778666)
Affinity DataKi:  367nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  387nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459074(Upamostat | Wx-671)
Affinity DataKi:  410nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529248(CHEMBL4547122)
Affinity DataKi:  439nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529252(CHEMBL4565975)
Affinity DataKi:  482nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529263(CHEMBL4438665)
Affinity DataKi:  499nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459064(CHEMBL4203547)
Affinity DataKi:  508nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529251(CHEMBL4554541)
Affinity DataKi:  578nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529244(CHEMBL4447661)
Affinity DataKi:  587nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  639nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529262(CHEMBL4575138)
Affinity DataKi:  642nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459077(CHEMBL4210813)
Affinity DataKi:  658nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565000(CHEMBL4791959)
Affinity DataKi:  688nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565000(CHEMBL4791959)
Affinity DataKi:  758nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529258(CHEMBL4451872)
Affinity DataKi:  771nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529253(CHEMBL4450051)
Affinity DataKi:  776nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459052(CHEMBL4211642)
Affinity DataKi:  884nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529249(CHEMBL4527266)
Affinity DataKi:  904nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459063(CHEMBL4218928)
Affinity DataKi:  934nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459057(CHEMBL4203367)
Affinity DataKi:  1.03E+3nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529255(CHEMBL4476829)
Affinity DataKi:  1.21E+3nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]-Ketanserin from human 5HT2A receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529254(CHEMBL4576924)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459058(CHEMBL4207061)
Affinity DataKi:  1.32E+3nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)
Affinity DataKi:  1.36E+3nMAssay Description:Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529259(CHEMBL4546029)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50529260(CHEMBL4551391)
Affinity DataKi:  1.48E+3nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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