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Found 25 with Last Name = 'covey' and Initial = 'df'
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM91718(Androst-1,4-dien-3,17-dione, 7)
Affinity DataKi:  120nMAssay Description:Inactivation rate (Ki) for human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit rho-3(Homo sapiens (Human))
University of Alabama At Birmingham

Curated by PDSP Ki Database
LigandPNGBDBM85712(1H-imidazol-4-ylacetic acid | CAS_645-65-8 | CHEMB...)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataKi:  220nMAssay Description:Competitive inhibition of binding to human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM91718(Androst-1,4-dien-3,17-dione, 7)
Affinity DataKi:  260nMAssay Description:Inactivation rate (Ki) for human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit rho-3(Homo sapiens (Human))
University of Alabama At Birmingham

Curated by PDSP Ki Database
LigandPNGBDBM81478(CAS_37539-03-0 | TACA)
Affinity DataKi:  360nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50014314(9a,11a-Dimethyl-3a,4,5,9a,9b,10,11,11a-octahydro-3...)
Affinity DataKi:  390nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50014314(9a,11a-Dimethyl-3a,4,5,9a,9b,10,11,11a-octahydro-3...)
Affinity DataKi:  410nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit rho-3(Homo sapiens (Human))
University of Alabama At Birmingham

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  460nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit rho-3(Homo sapiens (Human))
University of Alabama At Birmingham

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  580nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020640(10,13-Dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dod...)
Affinity DataKi:  690nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020640(10,13-Dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dod...)
Affinity DataKi:  1.10E+3nMAssay Description:Inactivation rate (Ki) for human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataKi:  1.55E+3nMAssay Description:Inactivation rate (Ki) for human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50406414(CHEMBL76061)
Affinity DataKi:  2.80E+3nMAssay Description:Tested by protection experiments to demonstrate the inactivation of estradiol dehydrogenase and the kinetic parameter Ki app was reported at a concen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020645(2,4b-Dimethyl-7-oxo-1,2,3,4,4a,4b,7,9,10,10a-decah...)
Affinity DataKi:  3.98E+3nMAssay Description:Inactivation rate (Ki) of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020647(7-Hydroxymethyl-4a,7-dimethyl-4b,5,6,7,8,8a,9,10-o...)
Affinity DataKi:  8.56E+3nMAssay Description:Inactivation rate (Ki) of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit rho-3(Homo sapiens (Human))
University of Alabama At Birmingham

Curated by PDSP Ki Database
LigandPNGBDBM50032955(1,2,3,6-Tetrahydro-pyridine-4-carboxylic acid | 1,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020641(Acetic acid 2,4b-dimethyl-7-oxo-1,2,3,4,4a,4b,7,9,...)
Affinity DataKi:  1.30E+4nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020639(7-Acetyl-4a,7-dimethyl-4b,5,6,7,8,8a,9,10-octahydr...)
Affinity DataKi:  4.50E+4nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50015834(CHEMBL307621 | Diastereomer-7-Methyl-7-(4,4,4-trif...)
Affinity DataKi:  5.90E+4nMAssay Description:Tested for time-dependent inactivation of the enzyme that followed pseudo- first- order kinetics in the absence of NAD+ and the Ki values were report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50015835(CHEMBL75893 | Diastereomer-7-Methyl-7-(4,4,4-trifl...)
Affinity DataKi:  6.50E+4nMAssay Description:Tested for time-dependent inactivation of the enzyme that followed pseudo- first- order kinetics in the absence of NAD+ and the Ki values were report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020642(4a,7-Dimethyl-7-propionyl-4b,5,6,7,8,8a,9,10-octah...)
Affinity DataKi:  9.70E+4nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020644(1,2,4b-Trimethyl-7-oxo-1,2,3,4,4a,4b,7,9,10,10a-de...)
Affinity DataKi:  1.03E+5nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020643(2,4b-Dimethyl-7-oxo-1,2,3,4,4a,4b,7,9,10,10a-decah...)
Affinity DataKi:  1.30E+5nMAssay Description:Competitive inhibition of binding to human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020638(2,4b-Dimethyl-7-oxo-1,2,3,4,4a,4b,7,9,10,10a-decah...)
Affinity DataKi:  8.93E+5nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50020646(1,2,4b-Trimethyl-7-oxo-1,2,3,4,4a,4b,7,9,10,10a-de...)
Affinity DataKi:  1.20E+6nMAssay Description:Competitive inhibition of binding to human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed