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Found 560 with Last Name = 'craig' and Initial = 'ra'
LigandPNGBDBM289504(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50609715(CHEMBL5286166)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609716(CHEMBL5272522)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609715(CHEMBL5286166)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002514(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609719(CHEMBL5283101)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50059190(CHEMBL3393333)
Affinity DataIC50:  3nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50609718(CHEMBL5288706)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50059190(CHEMBL3393333)
Affinity DataIC50:  3nMAssay Description:Inhibition of LZK (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50609708(CHEMBL5281494)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand InfoPDB
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002523(3-{6-[(6-Acetoxy-naphthalene-2-carbonyl)-amino]-2-...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002528(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609717(CHEMBL5271665)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609705(CHEMBL5268969)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609700(CHEMBL5271972)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002485(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002529(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609705(CHEMBL5268969)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609717(CHEMBL5271665)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609700(CHEMBL5271972)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002498(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002516(3-{6-[(6-Acetoxy-naphthalene-2-carbonyl)-amino]-2-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609714(CHEMBL5270353)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM289504(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of LZK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50609697(GDC-0134 | Gdc-0134 | Rg-6000)
Affinity DataIC50:  11nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609714(CHEMBL5270353)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609716(CHEMBL5272522)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609712(CHEMBL5276415)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609711(CHEMBL5268950)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609710(CHEMBL5276337)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002490(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  13nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609701(CHEMBL5277276)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609697(GDC-0134 | Gdc-0134 | Rg-6000)
Affinity DataIC50:  14nMAssay Description:Inhibition of LZK (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002484(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  14nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002504(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  14nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002519(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  15nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002521(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  16nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609708(CHEMBL5281494)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand InfoPDB
LigandPNGBDBM50609707(CHEMBL5284890)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002511(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  19nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50141730((2S,3R)-3-Amino-5-ethylsulfanyl-2-hydroxy-pentanoi...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against human methionine aminopeptidase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50141759((R)-3-Amino-2-hydroxy-5-phenyl-pentanoic acid ((S)...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against human methionine aminopeptidase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002483(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  21nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002501(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  22nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002481(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  22nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609712(CHEMBL5276415)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human LZK (9 to 114 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50609704(CHEMBL5278185)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50:  25nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50609703(CHEMBL5269484)
Affinity DataIC50:  28nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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