TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]DAMGO from MOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3H]U69593 from KOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation count...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor in mouse whole brain membrane measured after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
Affinity DataKi: 153nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 168nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 228nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 257nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 286nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 313nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
Affinity DataKi: 574nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 602nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 714nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Maryland
Curated by PDSP Ki Database
University of Maryland
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 790nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 793nMAssay Description:Displacement of [3H]U69593 from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 828nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair