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Found 112 with Last Name = 'dairaghi' and Initial = 'dj'
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL5/RANTES-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL15/Leukotactin1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427070(CHEMBL2322853)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL23/CKbeta8.1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  3.90nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL3/MIP-1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL15/Leukotactin1-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427105(CHEMBL2322879)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427095(CHEMBL2322858)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  5.5nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL3/MIP-1alpha-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427092(CHEMBL2322861)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427093(CHEMBL2322860)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427080(CHEMBL2322844)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427094(CHEMBL2322859)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427086(CHEMBL2322867)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427077(CHEMBL2322847)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427104(CHEMBL2322880)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427076(CHEMBL2321887)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427069(CHEMBL2322854)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427098(CHEMBL2322886)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427108(CHEMBL2322876)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CCL15/Leukotactin1 from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]-CCL15/Leukotactin1 from CCR1 in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427103(CHEMBL2322881)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183119(4-(((2-(trifluoromethyl)benzyl)(cyclohexylmethyl)a...)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at CCR1 in human monocytes assessed as inhibition of CCL15/Leukotactin1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427079(CHEMBL2322845)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427097(CHEMBL2322887)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183091(4-((bis(cyclohexylmethyl)amino)methyl)-N-(naphthal...)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427090(CHEMBL2322863)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427096(CHEMBL2322857)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427078(CHEMBL2322846)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427067(CHEMBL2322856)
Affinity DataIC50:  23nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183091(4-((bis(cyclohexylmethyl)amino)methyl)-N-(naphthal...)
Affinity DataIC50:  31nMAssay Description:Displacement of [125I]MDC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427071(CHEMBL2322852)
Affinity DataIC50:  37nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183102(CHEMBL205279 | N-(4-tert-butylthiazol-2-yl)-1-meth...)
Affinity DataIC50:  37nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427081(CHEMBL2322843)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183117(4-((diisobutylamino)methyl)-N-(naphthalen-1-yl)thi...)
Affinity DataIC50:  45nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427084(CHEMBL2322869)
Affinity DataIC50:  47nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427085(CHEMBL2322868)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427101(CHEMBL2322883)
Affinity DataIC50:  52nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427083(CHEMBL2322870)
Affinity DataIC50:  68nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427107(CHEMBL2322877)
Affinity DataIC50:  77nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183113(4-tert-butyl-N-(naphthalen-1-yl)oxazol-2-amine | C...)
Affinity DataIC50:  80nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183118(4-tert-butyl-N-(naphthalen-1-yl)thiazol-2-amine | ...)
Affinity DataIC50:  80nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427068(CHEMBL2322855)
Affinity DataIC50:  92nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427066(CHEMBL2322888)
Affinity DataIC50:  93nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL3/MIP-1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427074(CHEMBL2322849)
Affinity DataIC50:  97nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427120(CHEMBL2322890)
Affinity DataIC50:  98nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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