Affinity DataKi: 0.631nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -50.9kJ/mole EC50: 91nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 1.26nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 1.26nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 1.58nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nM ΔG°: -49.2kJ/mole EC50: 6.5nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 3.16nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 3.98nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 5.01nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 5.01nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -46.5kJ/mole EC50: 109nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -46.5kJ/mole EC50: 181nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 6.31nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 6.31nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -46.1kJ/mole EC50: 54nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -46.1kJ/mole EC50: 17.5nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 7.94nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 7.94nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -45.7kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -45.7kJ/mole EC50: 191nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 10nM ΔG°: -45.2kJ/mole EC50: 174nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 10nM ΔG°: -45.2kJ/mole EC50: 73nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Affinity DataKi: 10nM ΔG°: -45.2kJ/mole EC50: 9.60nMpH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Neuroscience Cedd Glaxosmithkline Research & Development
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to NK3 receptorMore data for this Ligand-Target Pair