TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of Eu-NDP-MSH from human MC1R expressed in HEK293T cells after 2 hrs by DELFIA methodMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells assessed as increase in accumulation of Hoechst 33342 preincubated for 30 mins followed by Hoechst...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.83E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.37E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 2.81E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.80nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.82E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 503nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.18E+4nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.96E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 620nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.25E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 640nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.68E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.17E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 164nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 0.350nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 0.0180nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.18E+3nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0300nMAssay Description:Agonist activity at mouse melanocortin 5 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 85nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 780nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 650nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.140nMAssay Description:Agonist activity at mouse melanocortin 3 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.73E+3nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.06E+3nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.21E+3nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 495nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.190nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0700nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.150nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair