TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for nicotinic acetylcholine receptor alpha 7 from human neuroblastoma SH-SY5Y cells; n=3More data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 1.46E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 1.55E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.27E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.66E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.77E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:Binding affinity for nicotinic acetylcholine receptor alpha 7 from human neuroblastoma SH-SY5Y cells; n=3More data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity for nicotinic acetylcholine receptor alpha 7 from human neuroblastoma SH-SY5Y cells; n=3More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.38E+5nMAssay Description:Binding affinity for nicotinic acetylcholine receptor alpha 7 from human neuroblastoma SH-SY5Y cells; n=3More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of Fibrinogen ReceptorMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 218nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 257nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 795nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair