Affinity DataIC50: <10nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: <10nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: <10nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development
Curated by ChEMBL
Novo Nordisk Research And Development
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cells in presence of 2 mM ATPMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 92nMAssay Description:Receptor binding affinity of the compound to human Peroxisome proliferator activated receptor gamma against [3H]-ragalitazar radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Compound was tested to inhibit lipoprotein lipase (LPL)More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibitory concentration against butyrylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of hormone sensitive lipase (HSL).More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human hormone-sensitive lipaseMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development
Curated by ChEMBL
Novo Nordisk Research And Development
Curated by ChEMBL
Affinity DataIC50: 286nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cells in presence of 2 mM ATPMore data for this Ligand-Target Pair