Compile Data Set for Download or QSAR
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Found 151 with Last Name = 'espitia' and Initial = 'sa'
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056605(7-Chloro-6-methyl-5-nitro-1,4-dihydro-quinoxaline-...)
Affinity DataIC50:  4.70nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091637(5-(3-(4-benzylpiperidin-1-yl)prop-1-ynyl)-1H-benzo...)
Affinity DataIC50:  5.30nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50038161(6,7-Dichloro-3-hydroxy-5-nitro-3,4-dihydro-1H-quin...)
Affinity DataIC50:  5.90nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091635(5-{3-[4-(3-Fluoro-benzyl)-piperidin-1-yl]-prop-1-y...)
Affinity DataIC50:  6.10nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091636(5-{3-[4-(4-Fluoro-benzyl)-piperidin-1-yl]-prop-1-y...)
Affinity DataIC50:  8.20nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056596(7-Bromo-6-methyl-5-nitro-1,4-dihydro-quinoxaline-2...)
Affinity DataIC50:  8.70nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091647(5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1,3-di...)
Affinity DataIC50:  16nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091632(5-{3-[4-(4-Methyl-benzyl)-piperidin-1-yl]-prop-1-y...)
Affinity DataIC50:  17nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091643(5-{3-[4-(4-Chloro-benzyl)-piperidin-1-yl]-prop-1-y...)
Affinity DataIC50:  19nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091626(5-[3-(4-Benzyl-4-hydroxy-piperidin-1-yl)-prop-1-yn...)
Affinity DataIC50:  19nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056618(6,7-Dibromo-5-nitro-1,4-dihydro-quinoxaline-2,3-di...)
Affinity DataIC50:  20nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091629(5-{3-[4-(4-Fluoro-benzyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataIC50:  24nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50079386(4-[2-(4-Benzyl-piperidin-1-yl)-ethoxy]-phenol | 4-...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091628(5-{3-[4-(4-Methoxy-benzyl)-piperidin-1-yl]-prop-1-...)
Affinity DataIC50:  26nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50079389(4-{2-[4-(4-Methyl-benzyl)-piperidin-1-yl]-ethoxy}-...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056620(6-Chloro-7-ethyl-5-nitro-1,4-dihydro-quinoxaline-2...)
Affinity DataIC50:  29nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056595(6,7-Dimethyl-5-nitro-1,4-dihydro-quinoxaline-2,3-d...)
Affinity DataIC50:  29nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50079385(1-[2-(4-Hydroxy-phenoxy)-ethyl]-4-(4-methyl-benzyl...)
Affinity DataIC50:  43nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056600(6-Chloro-7-methyl-5-nitro-1,4-dihydro-quinoxaline-...)
Affinity DataIC50:  45nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091645(6-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-3H-ben...)
Affinity DataIC50:  49nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50079388(4-{2-[4-(4-Fluoro-benzyl)-piperidin-1-yl]-ethoxy}-...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056591(7-Bromo-6-methoxy-5-nitro-1,4-dihydro-quinoxaline-...)
Affinity DataIC50:  64nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056598(7-Methyl-8-nitro-2,3-dioxo-1,2,3,4-tetrahydro-quin...)
Affinity DataIC50:  73nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056611(6-Bromo-7-ethyl-5-nitro-1,4-dihydro-quinoxaline-2,...)
Affinity DataIC50:  82nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091627(5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1,3-dih...)
Affinity DataIC50:  89nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056597(7-Fluoro-6-methyl-5-nitro-1,4-dihydro-quinoxaline-...)
Affinity DataIC50:  95nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091649(6-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1-meth...)
Affinity DataIC50:  98nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2B NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50078498(4-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-phenol...)
Affinity DataIC50:  100nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB N-methyl-D-aspartate (NMDA) expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50007674((+)-erythro 4-[2-(4-Benzyl-piperidin-1-yl)-1-hydro...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091634(5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1,3-di...)
Affinity DataIC50:  110nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091642(6-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-3H-benz...)
Affinity DataIC50:  120nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM22778(6,7-Dichloro-1,4-dihydro-quinoxaline-2,3-dione | 6...)
Affinity DataIC50:  130nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056592(7-Chloro-6-ethyl-5-nitro-1,4-dihydro-quinoxaline-2...)
Affinity DataIC50:  130nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056615(5-Amino-7-chloro-6-methyl-1,4-dihydro-quinoxaline-...)
Affinity DataIC50:  150nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056621(7-Chloro-6-methoxy-5-nitro-1,4-dihydro-quinoxaline...)
Affinity DataIC50:  150nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056606(6,7-Diethyl-5-nitro-1,4-dihydro-quinoxaline-2,3-di...)
Affinity DataIC50:  160nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50078480(4-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-phenol ...)
Affinity DataIC50:  170nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB N-methyl-D-aspartate (NMDA) expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091633(5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1,3-dih...)
Affinity DataIC50:  180nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091640(5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1H-benz...)
Affinity DataIC50:  220nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091648(5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1H-inda...)
Affinity DataIC50:  250nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091644(5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1,3-dih...)
Affinity DataIC50:  320nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091641(5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1H-ind...)
Affinity DataIC50:  380nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091639(5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1H-ben...)
Affinity DataIC50:  420nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB NMDA expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50048173(C,C,C-Trifluoro-N-(7-nitro-2-oxo-1,2-dihydro-quino...)
Affinity DataIC50:  620nMAssay Description:Inhibition of binding of [3H]-DCKA to N-methyl-D-aspartate glutamate receptor 1 in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50091625(5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1H-indo...)
Affinity DataIC50:  630nMAssay Description:Concentration required for 50% Inhibition of responses at cloned NR1A/2AB N-methyl-D-aspartate (NMDA) expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50079390(4-Benzyl-1-(2-phenoxy-ethyl)-piperidine | CHEMBL10...)
Affinity DataIC50:  630nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056593(7-Chloro-6-ethylsulfanyl-5-nitro-1,4-dihydro-quino...)
Affinity DataIC50:  640nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50060699(7-Nitro-5-oxy-1,4-dihydro-pyrido[2,3-b]pyrazine-2,...)
Affinity DataIC50:  690nMAssay Description:Binding affinity in rat brain cortical membranes by the displacement of [3H]- DCKA at N-methyl-D-aspartate glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50056622(6-Chloro-7-methyl-1,4-dihydro-quinoxaline-2,3-dion...)
Affinity DataIC50:  780nMAssay Description:Potency for the N-methyl-D-aspartate glutamate receptor 1 glycine site by displacement of [3H]5,7-dichlorokynurenic acid (DCKA) binding in rat brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50060694(7-Bromo-5-oxy-1,4-dihydro-pyrido[2,3-b]pyrazine-2,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity in rat brain cortical membranes by the displacement of [3H]- DCKA at N-methyl-D-aspartate glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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